SCHEMBL10077296

SCHEMBL10077296

CN(Cc1ccc(F)cc1-n1cncn1)C(=O)c1nc2n(c(=O)c1O)CCN2Cc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CLPP Q16740 8/20 0.37
ALDH1A1 P00352 2/20 0.34
LMNA P02545 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
HSD17B10 Q99714 1/20 0.34
PKM P14618 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
ATM Q13315 2/20 0.33
POLB P06746 1/20 0.33
NAMPT P43490 1/20 0.33
TP53 P04637 1/20 0.32
PLA2G7 Q13093 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4392728 0.85 CLPP (0.38) CLPPALDH1A1LMNASMN1; SMN2KDM4E
SCHEMBL4392377 0.76 CLPP (0.36) CLPPALDH1A1LMNASMN1; SMN2KDM4E
SCHEMBL4393723 0.73 CYP2C9 (0.36) ALDH1A1KDM4E
SCHEMBL4401303 0.73 CYP2C9 (0.36) TP53
SCHEMBL4398133 0.73 CYP2C9 (0.36)
SCHEMBL4397400 0.73 MAPK8 (0.36) PLA2G7
SCHEMBL4399670 0.70 SCD (0.43) CLPPALDH1A1LMNASMN1; SMN2KDM4E
SCHEMBL4397223 0.70 CYP2C9 (0.37)
SCHEMBL4403363 0.69 F2 (0.34) CLPPLMNATSHR
SCHEMBL4393694 0.69 FNTA (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919921-B1 BICYCLIC HETEROCYCLES AS HIV INTEGRASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2012-06-27 EP disclosed