SCHEMBL1007741

SCHEMBL1007741

CC(C)(C)[Si](C)(C)OCC1COCCN1c1nc2c(C(=O)O)cccc2o1.[LiH]

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 19/20 0.49
KCNH2 Q12809 3/20 0.40
CYP2C19 P33261 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1008074 0.99 HTR3A (0.50) HTR3AKCNH2CYP2C19NPC1RAB9A
SCHEMBL1008075 0.99 HTR3A (0.50) HTR3AKCNH2CYP2C19NPC1RAB9A
Lithium Ion SCHEMBL1007740 0.91 HTR3A (0.49) HTR3AKCNH2CYP2C19
SCHEMBL1007163 0.90 HTR3A (0.51) HTR3AKCNH2
SCHEMBL1007165 0.90 HTR3A (0.51) HTR3AKCNH2
SCHEMBL1006017 0.83 HTR3A (0.66) HTR3AKCNH2
SCHEMBL1004970 0.83 HTR3A (0.66) HTR3AKCNH2
SCHEMBL1004971 0.83 HTR3A (0.66) HTR3AKCNH2
SCHEMBL1005124 0.82 HTR3A (0.78) HTR3AKCNH2CYP2C19
SCHEMBL1007050 0.82 HTR3A (0.67) HTR3AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7863271-B2 2-aminobenzoxazole carboxamides as 5HT3 modulators ALBANY MOLECULAR RESEARCH, INC. (US) 2011-01-04 US disclosed