SCHEMBL10080435

SCHEMBL10080435

Cn1c(=O)c(C(N)=O)c(O)c2sccc21

nearest known ligand 0.62

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 1/20 0.62
FEN1 P39748 12/20 0.40
ALDH1A1 P00352 1/20 0.40
ERCC5 P28715 7/20 0.40
KCNH2 Q12809 1/20 0.39
EGFR P00533 1/20 0.37
SRC P12931 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3634507 0.86 EGLN1 (0.67) EGLN1FEN1ERCC5
SCHEMBL30041054 0.82 EGLN1 (0.63) EGLN1FEN1ALDH1A1ERCC5KCNH2
SCHEMBL2500134 0.79 EGLN1 (0.66) EGLN1FEN1ERCC5KCNH2
SCHEMBL2497674 0.79 ALDH1A1 (0.61) EGLN1FEN1ALDH1A1
SCHEMBL2493231 0.77 EGLN1 (1.00) EGLN1KCNH2
SCHEMBL14034795 0.76 EGLN1 (0.72) EGLN1FEN1ERCC5KCNH2
SCHEMBL4492683 0.76 MEN1 (0.66) EGLN1FEN1ALDH1A1ERCC5KCNH2
SCHEMBL2496618 0.75 EGLN1 (0.78) EGLN1KCNH2
SCHEMBL29079643 0.73 EGLN1 (0.49) EGLN1FEN1ALDH1A1ERCC5
SCHEMBL35212365 0.72 ALDH1A1 (0.74) ALDH1A1EGFRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150251-B9 THIENOPYRIDINE AND THIAZOLOPYRIDINE DERIVATIVES THAT INHIBIT PROLYL HYDROXYLASE ACTIVITY AMGEN INC (US) 2013-02-27 EP disclosed
EP-2150251-B1 THIENOPYRIDINE AND THIAZOLOPYRIDINE DERIVATIVES THAT INHIBIT PROLYL HYDROXYLASE ACTIVITY AMGEN INC (US) 2012-06-27 EP disclosed