SCHEMBL10080449

SCHEMBL10080449

CCCCCc1ccc2nc(C(=O)O)ccc2c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
MEN1 O00255 2/20 0.52
MAPT P10636 2/20 0.52
KMT2A Q03164 2/20 0.52
KDM4E B2RXH2 1/20 0.52
LMNA P02545 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
PKM P14618 1/20 0.52
ALOX15 P16050 1/20 0.52
TSHR P16473 1/20 0.52
NFKB1 P19838 1/20 0.52
THPO P40225 1/20 0.52
BLM P54132 1/20 0.52
PMP22 Q01453 1/20 0.52
HIF1A Q16665 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
KAT8 Q9H7Z6 2/20 0.50
PPARA Q07869 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6290855 0.79 TLR8 (0.54) ALDH1A1KDM4ELMNACYP3A4HIF1A
SCHEMBL13536956 0.78 PKM (0.39) ALDH1A1MEN1MAPTKMT2AKDM4E
SCHEMBL6289604 0.77 TLR8 (0.55) ALDH1A1MAPTKDM4ELMNACYP3A4
SCHEMBL15045025 0.77 MGAM (0.51) ALDH1A1MEN1MAPTKMT2AKDM4E
SCHEMBL11054926 0.77 TP53 (0.54) TSHRRARB
SCHEMBL10081274 0.76 GRIN2D (0.68) ALDH1A1MEN1MAPTKMT2ATSHR
SCHEMBL28065707 0.76 TLR8 (0.53) ALDH1A1KDM4ELMNACYP1A2CYP3A4
SCHEMBL23674307 0.76 OXER1 (0.45) ALDH1A1KAT8PPARATLR8PPARG
SCHEMBL9295912 0.75 MGAM (0.46) ALDH1A1MEN1MAPTKMT2AKDM4E
SCHEMBL7331987 0.75 GRIN2D (0.67) ALDH1A1MEN1MAPTKMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012019106-A2 POSITIVE AND NEGATIVE MODULATORS OF NMDA RECEPTORS BOARD OF REGENTS OF THE UNIVERSITY OF NEBRASKA (US) 2012-02-09 WO disclosed