SCHEMBL10083019

SCHEMBL10083019

O=C(NC(CN1CCCC1)c1ccccc1)C1(c2cnc3ccccc3c2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 1/20 0.48
ITGB7 P26010 1/20 0.48
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GPR88 Q9GZN0 1/20 0.40
RPS6KB1 P23443 2/20 0.39
AURKA O14965 1/20 0.39
AURKB Q96GD4 1/20 0.39
TRPV1 Q8NER1 2/20 0.39
MITF O75030 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HTT P42858 1/20 0.39
GFER P55789 1/20 0.39
PAX8 Q06710 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10083317 1.00 ITGA4 (0.48) ITGA4ITGB7ROCK2ROCK1RAB9A
Hydrochloric Acid SCHEMBL434712 0.99 ITGA4 (0.47) ITGA4ITGB7ROCK2ROCK1RAB9A
Hydrochloric Acid SCHEMBL434711 0.99 ITGA4 (0.47) ITGA4ITGB7ROCK2ROCK1RAB9A
SCHEMBL433726 0.88 ITGA4 (0.47) ITGA4ITGB7RPS6KB1AKR1C3AKR1C2
SCHEMBL433725 0.88 ITGA4 (0.47) ITGA4ITGB7RPS6KB1AKR1C3AKR1C2
SCHEMBL435949 0.87 ITGA4 (0.44) ITGA4ITGB7AKR1C3AKR1C2FAAH
SCHEMBL434432 0.87 ITGA4 (0.44) ITGA4ITGB7AKR1C3AKR1C2FAAH
SCHEMBL15385502 0.87 ITGA4 (0.44) ITGA4ITGB7CNR2
SCHEMBL434349 0.87 ITGA4 (0.44) ITGA4ITGB7CNR2
SCHEMBL434182 0.87 ITGA4 (0.47) ITGA4ITGB7RPS6KB1AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012410-A2 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES LTD. (IN) 2012-01-26 WO disclosed