SCHEMBL10086642

SCHEMBL10086642

Fc1ccc(CNc2nc(Nc3cnccn3)cc(-c3ccccn3)n2)cc1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
HPGD P15428 2/20 0.55
KDM4E B2RXH2 1/20 0.55
GPR39 O43194 12/20 0.53
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
KCNH3 Q9ULD8 2/20 0.44
F2 P00734 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10086623 0.85 ALDH1A1 (0.55) ALDH1A1HPGDKDM4EF2
SCHEMBL10086635 0.85 ALDH1A1 (0.57) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL10086733 0.84 ALDH1A1 (0.57) ALDH1A1HPGDKDM4EGPR39MEN1
SCHEMBL10086735 0.82 KDM4E (0.54) ALDH1A1HPGDKDM4EKCNH3
SCHEMBL10086710 0.81 ALDH1A1 (0.53) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL10086638 0.81 ALDH1A1 (0.61) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL10086666 0.81 ALDH1A1 (0.61) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL12140755 0.81 JAK2 (0.53) GPR39MEN1KMT2A
SCHEMBL16503794 0.81 ALDH1A1 (0.52) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL10086674 0.81 ALDH1A1 (0.52) ALDH1A1HPGDKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020786-A1 PHARMACEUTICAL COMPOSITION 日本新薬株式会社 (JP) 2012-02-16 WO disclosed
WO-2012020787-A1 MALIGNANT LYMPHOMA THERAPEUTIC AGENT 日本新薬株式会社 (JP) 2012-02-16 WO disclosed
WO-2012005299-A1 ROS TYROSINE KINASE INHIBITOR 日本新薬株式会社 (JP) 2012-01-12 WO disclosed
WO-2010090290-A1 AMINOPYRAZINE DERIVATIVE AND MEDICINE 日本新薬株式会社 (JP) 2010-08-12 WO disclosed