SCHEMBL1009348

SCHEMBL1009348

CCCCCCCCc1ccc(C(C)N)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.60
ESR1 P03372 2/20 0.55
ADRA2A P08913 2/20 0.55
ADORA3 P0DMS8 2/20 0.55
TACR2 P21452 2/20 0.55
SLC6A2 P23975 2/20 0.55
SLC6A4 P31645 2/20 0.55
SLC6A3 Q01959 2/20 0.55
KDM4E B2RXH2 1/20 0.55
ALDH1A1 P00352 1/20 0.55
LMNA P02545 1/20 0.55
SHBG P04278 1/20 0.55
TP53 P04637 1/20 0.55
CYP3A4 P08684 1/20 0.55
HSPD1 P10809 1/20 0.55
ADRB3 P13945 1/20 0.55
HTR2C P28335 1/20 0.55
HSPE1 P61604 1/20 0.55
HIF1A Q16665 1/20 0.55
TST Q16762 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1313200 1.00 HTR2A (0.60) HTR2AESR1ADRA2AADORA3TACR2
SCHEMBL9945668 1.00 HTR2A (0.60) HTR2AESR1ADRA2AADORA3TACR2
Hydrochloric Acid SCHEMBL11737570 0.98 HTR2A (0.58) HTR2AESR1ADRA2AADORA3TACR2
SCHEMBL19174795 0.98 HTR2A (0.57) HTR2AESR1ADRA2AADORA3TACR2
SCHEMBL29342921 0.92 HTR2A (0.50) HTR2AESR1ADRA2AADORA3TACR2
SCHEMBL11686889 0.92 HTR2A (0.50) HTR2AESR1ADRA2AADORA3TACR2
SCHEMBL29342569 0.92 HTR2A (0.50) HTR2AESR1ADRA2AADORA3TACR2
SCHEMBL30469503 0.86 HTR2A (0.62) HTR2AESR1ADRA2AADORA3TACR2
SCHEMBL6861225 0.86 HTR2A (0.62) HTR2AESR1ADRA2AADORA3TACR2
Hydrochloric Acid SCHEMBL27998571 0.86 HTR2A (0.62) HTR2AESR1ADRA2AADORA3TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2303250-A1 PAEDIATRIC COMPOSITIONS FOR TREATING1 MULTIPLE SCLEROSIS Novartis AG (CH) 2011-04-06 EP claimed
US-20140274897-A1 METHOD FOR PREVENTING AND TREATING DIABETES USING NEURTURIN EVOTEC INTERNATIONAL GMBH (DE) 2014-09-18 US disclosed
US-8772233-B2 Method for promoting regeneration of pancreatic beta-cells by administering neurturin EVOTEC INTERNATIONAL GMBH (DE) 2014-07-08 US disclosed
US-20130150293-A1 METHOD FOR PREVENTING AND TREATING DIABETES USING NEURTURIN DEVELOGEN AKTIENGESELLSCHAFT (DE) 2013-06-13 US disclosed
US-20110256113-A1 METHOD FOR PREVENTING AND TREATING DIABETES USING NEURTURIN EVOTEC INTERNATIONAL GMBH (DE) 2011-10-20 US disclosed
WO-2011080733-A1 DEPOT SYSTEMS COMPRISING GLATIRAMER OR A PHARMACOLOGICALLY ACCEPTABLE SALT THEREOF MAPI PHARMA LIMITED (IL) 2011-07-07 WO disclosed
EP-2303250-A1 PAEDIATRIC COMPOSITIONS FOR TREATING1 MULTIPLE SCLEROSIS Novartis AG (CH) 2011-04-06 EP disclosed
EP-2268603-A1 PROCESS FOR THE PREPARATION OF 2-AMINO-2- [2- (4-C3-C21-ALKYL-PHENYL)ETHYL]PROPANE-1, 3-DIOLS Novartis AG (CH) 2011-01-05 EP disclosed
US-20100158874-A1 Compositions and Methods for Treating Peripheral Vascular Diseases MOUNT SINAI HOSPITAL (CA) 2010-06-24 US disclosed
US-20090298771-A1 USE OF SECRETED PROTEIN PRODUCTS FOR PREVENTING AND TREATING PANCREATIC DISEASES AND/OR OBESITY AND/OR METABOLIC SYNDROME DEVELOGEN AKTIENGESELLSCHAFT (DE) 2009-12-03 US disclosed
US-20080241106-A1 Using nervous system protein to induce stem cell differentiation into pancreatic tissues; tissue engineering and repair; regenerative medicine; DEVELOGEN AKTIENGESELLSCHAFT (DE) 2008-10-02 US disclosed
EP-1971363-A1 COMBINATION TREATMENTS WITH GASTRIN AGONISTS FOR DIABETES AND RELATED DISEASES Waratah Pharmaceuticals, Inc. (CA) 2008-09-24 EP disclosed
WO-2008104064-A1 COMPOSITIONS AND METHODS FOR TREATING PERIPHERAL VASCULAR DISEASES MOUNT SINAI HOSPITAL (CA) 2008-09-04 WO disclosed
WO-2008104065-A1 NEURAL CELL PREPARATIONS AND METHODS OF MAKING AND USING THEM MOUNT SINAI HOSPITAL (CA) 2008-09-04 WO disclosed
WO-2007062531-A1 COMBINATION TREATMENTS WITH GASTRIN AGONISTS FOR DIABETES AND RELATED DISEASES WARATAH PHARMACEUTICALS, INC. (CA) 2007-06-07 WO disclosed
US-20070110728-A1 Method for preventing and treating diabetes using dg119 DEVELOGEN AKTIENGESELLSCHAFT (DE) 2007-05-17 US disclosed
US-5948820-A IMMUNOSUPPRESSANT; PREVENT REJECTION OF ORGAN TRANSPLANT;AUTOIMMUNE DISEASES; MULTIPLE SCLEROSIS; LUPUS; ANTIALLERGENS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1999-09-07 US disclosed