SCHEMBL1009759

SCHEMBL1009759

CON=C(C(N)=O)c1ccccc1Oc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.50
RAB9A P51151 1/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
HTT P42858 1/20 0.46
MAPK1 P28482 1/20 0.45
NPSR1 Q6W5P4 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
PARP10 Q53GL7 1/20 0.42
ALDH1A1 P00352 3/20 0.42
TSHR P16473 3/20 0.42
GAA P10253 1/20 0.42
KDM4E B2RXH2 1/20 0.42
TTR P02766 1/20 0.42
SCN1A P35498 1/20 0.42
SCN2A Q99250 1/20 0.42
SCN3A Q9NY46 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8368445 1.00 CTNNB1 (0.59) CTNNB1SMN1; SMN2RAB9AMEN1KMT2A
SCHEMBL5079797 1.00 CTNNB1 (0.59) CTNNB1SMN1; SMN2RAB9AMEN1KMT2A
SCHEMBL8761574 0.88 CTNNB1 (0.54) CTNNB1SMN1; SMN2RAB9AMEN1KMT2A
SCHEMBL8761579 0.88 CTNNB1 (0.54) CTNNB1SMN1; SMN2RAB9AMEN1KMT2A
SCHEMBL10433687 0.87 ALDH1A1 (0.49) CTNNB1SMN1; SMN2RAB9AMEN1KMT2A
SCHEMBL10433688 0.87 ALDH1A1 (0.49) CTNNB1SMN1; SMN2RAB9AMEN1KMT2A
SCHEMBL9193371 0.85 CTNNB1 (0.51) CTNNB1SMN1; SMN2RAB9AMEN1KMT2A
SCHEMBL8343946 0.85 HIF1A (0.53) CTNNB1SMN1; SMN2RAB9AMEN1KMT2A
SCHEMBL8761257 0.85 HIF1A (0.53) CTNNB1SMN1; SMN2RAB9AMEN1KMT2A
SCHEMBL9196461 0.85 HIF1A (0.53) CTNNB1SMN1; SMN2RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-8231310-A None JP disclosed
JP-3246268-A None JP disclosed
JP-8253449-A None JP disclosed
EP-2268145-A1 METHOD OF PLANT GROWTH PROMOTION USING AMIDE COMPOUNDS Bayer CropScience AG (DE) 2011-01-05 EP disclosed
EP-1761498-A1 1-METHYL-3-DIFLUOROMETHYL-PYRAZOL-4-CARBONIC ACID-(ORTHO-PHENYL)-ANILIDES, AND USE THEREOF AS A FUNGICIDE BASF AKTIENGESELLSCHAFT (DE) 2007-03-14 EP disclosed
EP-1761499-A1 1-METHYL-3-TRIFLUOROMETHYL-PYRAZOLE-4-CARBOXYLIC ACID (ORTHO-PHENYL)-ANILIDES AND TO USE THEREOF AS FUNGICIDE BASF AKTIENGESELLSCHAFT (DE) 2007-03-14 EP disclosed
EP-1699763-A1 3-TRIFLUOROMETHYL PICOLINIC ACID ANILIDES, AND USE THEREOF AS FUNGICIDES BASF AKTIENGESELLSCHAFT (DE) 2006-09-13 EP disclosed
EP-1699752-A1 (HETERO)CYCLYL CARBOXANILIDES FOR CONTROLLING HARMFUL FUNGI BASF AKTIENGESELLSCHAFT (DE) 2006-09-13 EP disclosed
WO-2005123689-A1 1-METHYL-3-TRIFLUOROMETHYL-PYRAZOLE-4-CARBOXYLIC ACID (ORTHO-PHENYL)-ANILIDES AND TO USE THEREOF AS FUNGICIDE BASF AKTIENGESELLSCHAFT (DE) 2005-12-29 WO disclosed
WO-2005123690-A1 1-METHYL-3-DIFLUOROMETHYL-PYRAZOL-4-CARBONIC ACID-(ORTHO-PHENYL)-ANILIDES, AND USE THEREOF AS A FUNGICIDE BASF AKTIENGESELLSCHAFT (DE) 2005-12-29 WO disclosed
US-5371223-A Controlling phytopathogens SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-12-06 US disclosed
US-5371222-A Intermediates SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-12-06 US disclosed
US-5360810-A APPLYING TO PLANTS SHIONOGI & CO., LTD. (JP) 1994-11-01 US disclosed
EP-0617011-A2 Process for producing alkoxyiminoacetamide compounds SHIONOGI & CO., LTD. (JP) 1994-09-28 EP disclosed
EP-0596692-A2 A process for producing (E)-alkoxyimino or hydroxyiminoacetamide compounds and intermediates therefor SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-05-11 EP disclosed
US-5248687-A PHENYLMETHOXYIMINO COMPOUNDS AND AGRICULTURAL FUNGICIDES CONTAINING THEM SHIONOGI & CO., LTD. (JP) 1993-09-28 US disclosed
EP-0528681-A1 Phenylmethoxyimino compounds and agricultural fungicides containing them SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1993-02-24 EP disclosed
US-5185342-A ALKOXYIMINOACETAMIDE DERIVATIVES AND THEIR USE AS FUNGICIDES SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1993-02-09 US disclosed
JP-H03246268-A ALKOXYIMINOACETIC ACID AMIDE COMPOUND AND FUNGICIDE FOR AGRICULTURAL USE SHIONOGI & CO LTD 1991-11-01 JP disclosed
EP-0398692-A2 Alkoxyiminoacetamide derivatives and their use as fungicides SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1990-11-22 EP disclosed