SCHEMBL10104693

SCHEMBL10104693

C=C1c2[nH]cnc2NC(=O)N1CC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
GLA P06280 1/20 0.38
HPGD P15428 1/20 0.38
HIF1A Q16665 1/20 0.38
GDA Q9Y2T3 1/20 0.37
ADORA2A P29274 10/20 0.36
ADORA2B P29275 7/20 0.36
PDE4A P27815 9/20 0.35
PDE4B Q07343 9/20 0.35
PDE4C Q08493 9/20 0.35
PDE4D Q08499 9/20 0.35
MAPK14 Q16539 3/20 0.33
ATIC P31939 1/20 0.33
GMNN O75496 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
THPO P40225 1/20 0.31
BLM P54132 1/20 0.31
PMP22 Q01453 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12413543 0.74 GDA (0.34) ALDH1A1GDAADORA2BATIC
SCHEMBL15759316 0.65 GDA (0.39) ALDH1A1GDAATIC
SCHEMBL13771834 0.65 ATIC (0.47) ALDH1A1GDAATIC
SCHEMBL662729 0.62 GDA (0.40) ALDH1A1GDAATIC
SCHEMBL19090547 0.61 SMN1; SMN2 (0.38) ALDH1A1KDM4ELMNAMAPT
SCHEMBL13753310 0.59 F2 (0.42) ALDH1A1KDM4EGLAHPGDHIF1A
SCHEMBL17210366 0.58 MEN1 (0.33) ALDH1A1HIF1AADORA2AADORA2BPDE4A
SCHEMBL20656217 0.58 MEN1 (0.33) ALDH1A1HIF1AADORA2AADORA2BPDE4A
SCHEMBL15414257 0.57 GDA (0.42) ALDH1A1GDAATIC
SCHEMBL14154963 0.57 F2 (0.40) ALDH1A1KDM4EGLAHPGDHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2465859-A1 8-Triazolylxanthine derivatives, processes for their production and their use as adenosine receptor antagonists Life & Brain GmbH (DE) 2012-06-20 EP disclosed