SCHEMBL1010868

SCHEMBL1010868

CC1c2cccc(OC(=O)N(C)C)c2CCN1C(=O)c1cc2ncc(Cl)cn2n1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 7/20 0.41
ACHE P22303 4/20 0.41
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
ALDH1A1 P00352 2/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
ESR1 P03372 1/20 0.34
POLB P06746 1/20 0.34
ESR2 Q92731 1/20 0.34
STAT3 P40763 1/20 0.34
MGLL Q99685 1/20 0.34
F11 P03951 1/20 0.34
KLKB1 P03952 1/20 0.34
QRFPR Q96P65 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1011687 0.90 GRM5 (0.46) GRM5ACHEALDH1A1LMNAHPGD
SCHEMBL1010530 0.85 GRM5 (0.43) GRM5ALDH1A1LMNAHPGDESR1
SCHEMBL1009118 0.85 GRM5 (0.46) GRM5ALDH1A1LMNAHPGDESR1
SCHEMBL1010766 0.84 GRM5 (0.46) GRM5ALDH1A1LMNAHPGDESR1
SCHEMBL1010423 0.84 GRM5 (0.48) GRM5ALDH1A1LMNAHPGDESR1
SCHEMBL1013119 0.84 GRM5 (0.44) GRM5ALDH1A1LMNAHPGDPOLB
SCHEMBL1010289 0.83 GRM5 (0.45) GRM5ALDH1A1LMNAHPGDESR1
SCHEMBL4081280 0.83 GRM5 (0.44) GRM5ALDH1A1LMNAHPGDESR1
SCHEMBL1012541 0.83 GRM5 (0.44) GRM5ALDH1A1LMNAHPGDESR1
SCHEMBL1011045 0.82 GRM5 (0.43) GRM5ALDH1A1LMNAHPGDESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054416-B1 SUBSTITUTED PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO KGAA (DE) 2011-01-05 EP claimed