SCHEMBL10113675

SCHEMBL10113675

COC(=O)c1cccc(OCC2CCN(c3ccc(NC(=O)c4ccc5c(c4)OCCO5)cn3)CC2)c1

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 16/20 0.66
SOAT1 P35610 2/20 0.66
CYP3A4 P08684 1/20 0.66
SOAT2 O75908 1/20 0.54
DGAT2 Q96PD7 1/20 0.54
NPC1 O15118 3/20 0.52
RAB9A P51151 3/20 0.52
PKM P14618 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10113648 0.87 DGAT1 (0.85) DGAT1SOAT1CYP3A4SOAT2DGAT2
SCHEMBL10113683 0.87 DGAT1 (0.85) DGAT1SOAT1CYP3A4SOAT2DGAT2
SCHEMBL10113657 0.86 DGAT1 (0.86) DGAT1SOAT1CYP3A4SOAT2DGAT2
SCHEMBL10113677 0.85 DGAT1 (0.67) DGAT1SOAT1CYP3A4SOAT2DGAT2
SCHEMBL10113362 0.84 DGAT1 (0.78) DGAT1SOAT1CYP3A4SOAT2DGAT2
SCHEMBL10113637 0.84 DGAT1 (0.69) DGAT1SOAT1CYP3A4SOAT2DGAT2
SCHEMBL10113795 0.84 DGAT1 (0.77) DGAT1SOAT1CYP3A4SOAT2DGAT2
SCHEMBL10113678 0.83 DGAT1 (0.87) DGAT1SOAT1CYP3A4SOAT2DGAT2
SCHEMBL10113332 0.81 DGAT1 (0.86) DGAT1SOAT1CYP3A4SOAT2DGAT2
SCHEMBL10113656 0.80 DGAT1 (0.85) DGAT1SOAT1CYP3A4SOAT2DGAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012024179-A1 SUBSTITUTED AMIDE DERIVATIVES AS DGAT-1 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-02-23 WO disclosed