SCHEMBL1011758

SCHEMBL1011758

Cc1ccc(/C=C2\CCN(C(=O)O)C(C(C)(C)C)C2)cc1Oc1ccc(C(F)(F)F)cn1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.44
CYP2D6 P10635 4/20 0.44
FAAH O00519 16/20 0.42
GABRA1 P14867 1/20 0.41
ADRA2C P18825 1/20 0.41
CNR1 P21554 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
CNR2 P34972 1/20 0.41
HTR2B P41595 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1011760 1.00 CYP3A4 (0.44) CYP3A4CYP2D6FAAHGABRA1ADRA2C
SCHEMBL2543044 0.86 CYP3A4 (0.55) CYP3A4CYP2D6FAAHGABRA1ADRA2C
SCHEMBL1011759 0.81 CYP3A4 (0.52) CYP3A4CYP2D6FAAHGABRA1ADRA2C
SCHEMBL1009417 0.76 CYP3A4 (0.48) CYP3A4CYP2D6FAAHGABRA1ADRA2C
SCHEMBL1009415 0.76 CYP3A4 (0.48) CYP3A4CYP2D6FAAHGABRA1ADRA2C
SCHEMBL1012025 0.76 FAAH (0.51) CYP3A4CYP2D6FAAHGABRA1ADRA2C
SCHEMBL1011197 0.75 FAAH (0.44) CYP3A4CYP2D6FAAHCYP2C9
SCHEMBL1009793 0.73 CYP3A4 (0.76) CYP3A4CYP2D6FAAHGABRA1ADRA2C
SCHEMBL1010705 0.72 FAAH (0.50) CYP3A4CYP2D6FAAHGABRA1ADRA2C
SCHEMBL1010255 0.71 FAAH (0.43) CYP3A4CYP2D6FAAHGABRA1ADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2076508-B1 BIARYL ETHER UREA COMPOUNDS PFIZER PROD INC (US) 2011-01-05 EP disclosed