SCHEMBL10119686

SCHEMBL10119686

CC(C)NC(=O)N1CCC[C@H]1C(=O)Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3C(=O)N(C)C(C)C)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
CCR1 P32246 1/20 0.47
ALDH1A1 P00352 2/20 0.45
LMNA P02545 2/20 0.45
POLB P06746 1/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
MAPK1 P28482 1/20 0.44
TSHR P16473 1/20 0.44
KCNH2 Q12809 1/20 0.43
F2 P00734 2/20 0.42
PRSS1 P07477 2/20 0.42
PRSS2 P07478 2/20 0.42
PRSS3 P35030 2/20 0.42
NPC1 O15118 1/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL844894 0.91 CYP2C19 (0.55) CYP2C9CYP2C19ALDH1A1LMNAPOLB
SCHEMBL845202 0.86 CYP2C19 (0.48) CYP2C9CYP2C19ALDH1A1LMNAPOLB
SCHEMBL845488 0.86 CYP2C19 (0.48) CYP2C9CYP2C19ALDH1A1LMNAPOLB
SCHEMBL845759 0.86 CYP2C19 (0.48) CYP2C9CYP2C19ALDH1A1LMNAPOLB
SCHEMBL845774 0.84 CYP2C19 (0.49) CYP2C9CYP2C19ALDH1A1LMNAPOLB
SCHEMBL844890 0.80 KCNH2 (0.51) CYP2C9CYP2C19ALDH1A1LMNAPOLB
SCHEMBL845203 0.79 CCR1 (0.47) CYP2C9CYP2C19CCR1ALDH1A1LMNA
SCHEMBL844902 0.77 ALDH1A1 (0.47) CYP2C9CYP2C19CCR1ALDH1A1LMNA
SCHEMBL845245 0.77 PTPN1 (0.50) CYP2C9CYP2C19ALDH1A1LMNAPOLB
SCHEMBL845258 0.76 MAPK1 (0.60) CYP2C9CYP2C19ALDH1A1LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed