SCHEMBL10120303

SCHEMBL10120303

Cc1cncc(Cl)c1N1CCN(C(=O)CNc2c(-c3ccc(N4CCOCC4)nc3)nc3cnccn23)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 7/20 0.45
KDM4E B2RXH2 6/20 0.45
CASP1 P29466 3/20 0.45
CASP7 P55210 3/20 0.45
ALDH1A1 P00352 2/20 0.45
HPGD P15428 2/20 0.45
HSD17B10 Q99714 2/20 0.45
RXFP1 Q9HBX9 1/20 0.44
MAPT P10636 5/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
TP53 P04637 1/20 0.42
ALOX15 P16050 1/20 0.41
ALOX5 P09917 1/20 0.41
BRD4 O60885 3/20 0.40
TRIM33 Q9UPN9 1/20 0.38
KDR P35968 2/20 0.38
ETV6 P41212 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
CNR2 P34972 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15179450 0.95 GAA (0.44) GAAKDM4ECASP1CASP7ALDH1A1
SCHEMBL10120304 0.92 KDM4E (0.45) GAAKDM4ECASP1CASP7ALDH1A1
SCHEMBL10120316 0.88 KDM4E (0.46) GAAKDM4ECASP1CASP7ALDH1A1
SCHEMBL10120111 0.88 KDM4E (0.45) GAAKDM4ECASP1CASP7ALDH1A1
SCHEMBL15179409 0.86 CNR2 (0.42) GAAKDM4EALDH1A1HPGDHSD17B10
SCHEMBL10120107 0.86 KDM4E (0.44) GAAKDM4ECASP1CASP7ALDH1A1
SCHEMBL10120099 0.85 ALOX5 (0.43) GAAMAPTTP53ALOX5BRD4
SCHEMBL15179298 0.83 GAA (0.48) GAAKDM4ECASP1CASP7ALDH1A1
SCHEMBL10120106 0.82 CNR2 (0.43) GAAKDM4EALDH1A1MAPTRAB9A
SCHEMBL15179269 0.82 GAA (0.47) GAAKDM4ECASP1CASP7ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012018662-A2 FUSED-IMIDAZOYL COMPOUNDS USEFUL AS ANTIMICROBIAL AGENTS SCHERING CORPORATION (US) 2012-02-09 WO disclosed