SCHEMBL10121020

SCHEMBL10121020

C=C1N[C@](CCC2CCCCC2)(C[C@H]2CCC[C@@H](NCc3cccnc3)C2)C(=O)N1C

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
PKM P14618 1/20 0.44
BACE1 P56817 15/20 0.44
CTSD P07339 13/20 0.44
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13475796 0.90 BACE1 (0.45) KDM4EALDH1A1PKMBACE1CTSD
SCHEMBL7538417 0.90 BACE1 (0.45) KDM4EALDH1A1PKMBACE1CTSD
SCHEMBL7538463 0.90 BACE1 (0.45) KDM4EALDH1A1PKMBACE1CTSD
SCHEMBL13475791 0.90 BACE1 (0.45) KDM4EALDH1A1PKMBACE1CTSD
SCHEMBL12174373 0.90 BACE1 (0.45) KDM4EALDH1A1PKMBACE1CTSD
SCHEMBL7538420 0.90 BACE1 (0.45) KDM4EALDH1A1PKMBACE1CTSD
SCHEMBL7534142 0.90 BACE1 (0.45) KDM4EALDH1A1PKMBACE1CTSD
SCHEMBL10121023 0.90 BACE1 (0.47) KDM4EBACE1CTSDGAA
SCHEMBL10121024 0.90 BACE1 (0.47) KDM4EBACE1CTSDGAA
SCHEMBL7533208 0.83 BACE1 (0.43) KDM4EALDH1A1PKMBACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178513-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-15 US disclosed