SCHEMBL10121023

SCHEMBL10121023

C=C1N[C@](CCC2CCCCC2)(C[C@H]2CCC[C@H](NCc3ccncc3)C2)C(=O)N1C

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 17/20 0.47
CTSD P07339 14/20 0.47
EPHX1 P07099 1/20 0.36
MAPT P10636 1/20 0.36
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10121024 1.00 BACE1 (0.47) BACE1CTSDEPHX1MAPTKDM4E
SCHEMBL10121020 0.90 KDM4E (0.44) BACE1CTSDKDM4EGAA
SCHEMBL8267582 0.90 BACE1 (0.47) BACE1CTSDEPHX1MAPTKDM4E
SCHEMBL7533157 0.90 BACE1 (0.47) BACE1CTSDEPHX1MAPTKDM4E
SCHEMBL7534839 0.90 BACE1 (0.47) BACE1CTSDEPHX1MAPTKDM4E
SCHEMBL7534011 0.90 BACE1 (0.47) BACE1CTSDEPHX1MAPTKDM4E
SCHEMBL8289262 0.90 BACE1 (0.47) BACE1CTSDEPHX1MAPTKDM4E
SCHEMBL7538661 0.90 BACE1 (0.47) BACE1CTSDEPHX1MAPTKDM4E
SCHEMBL10121004 0.83 BACE1 (0.46) BACE1CTSD
SCHEMBL10121006 0.82 BACE1 (0.44) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178513-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-15 US disclosed