SCHEMBL10124916

SCHEMBL10124916

Nc1nc(-c2ccnc3[nH]ccc23)nc2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 3/20 0.56
CHUK O15111 3/20 0.56
DAPK3 O43293 1/20 0.56
JAK2 O60674 1/20 0.56
PRKD3 O94806 1/20 0.56
MAP4K4 O95819 1/20 0.56
PAK4 O96013 1/20 0.56
CSF1R P07333 1/20 0.56
RET P07949 1/20 0.56
IGF1R P08069 1/20 0.56
FGFR1 P11362 1/20 0.56
PRKACA P17612 1/20 0.56
FLT1 P17948 1/20 0.56
LTK P29376 1/20 0.56
GRK5 P34947 1/20 0.56
KDR P35968 1/20 0.56
MAP2K2 P36507 1/20 0.56
MAPK8 P45983 1/20 0.56
CSNK1A1 P48729 1/20 0.56
CDK8 P49336 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16897104 0.85 LATS1 (0.61) IKBKBCHUKDAPK3JAK2PRKD3
SCHEMBL12127272 0.74 PRKCI (0.67) IKBKBCHUKDAPK3JAK2PRKD3
SCHEMBL29789047 0.74 PRKCI (0.67) IKBKBCHUKDAPK3JAK2PRKD3
SCHEMBL12346464 0.74 NUDT1 (0.57) IKBKBCHUKDAPK3JAK2PRKD3
SCHEMBL22160800 0.74 BRAF (0.57) IKBKBCHUKDAPK3JAK2PRKD3
SCHEMBL857275 0.73 IKBKB (1.00) IKBKBCHUKDAPK3JAK2PRKD3
SCHEMBL2097365 0.72 IKBKB (0.63) IKBKBCHUKDAPK3JAK2PRKD3
SCHEMBL2240671 0.72 AURKB (0.71) IKBKBCHUKDAPK3JAK2PRKD3
Hydrochloric Acid SCHEMBL11360576 0.71 CYP1A1 (0.50) CSNK1A1TYRO3DYRK1BCYP1A1CYP1A2
SCHEMBL14529392 0.71 CYP1A1 (0.54) CYP1A1CYP1A2CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881983-B1 PYRROLOPYRIDINES USEFUL AS INHIBITORS OF PROTEIN KINASE VERTEX PHARMA (US) 2012-01-11 EP disclosed