SCHEMBL10124969

SCHEMBL10124969

CNC(=O)c1ccc(-c2ccnc3[nH]ccc23)s1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 8/20 0.62
IKBKB O14920 2/20 0.46
CHUK O15111 2/20 0.46
KDM4E B2RXH2 2/20 0.46
NPC1 O15118 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
RAB9A P51151 2/20 0.46
NUDT1 P36639 2/20 0.45
NEK1 Q96PY6 1/20 0.44
AURKB Q96GD4 2/20 0.43
DAPK3 O43293 1/20 0.43
JAK2 O60674 1/20 0.43
PRKD3 O94806 1/20 0.43
MAP4K4 O95819 1/20 0.43
PAK4 O96013 1/20 0.43
CSF1R P07333 1/20 0.43
RET P07949 1/20 0.43
IGF1R P08069 1/20 0.43
FGFR1 P11362 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4791074 0.87 AKT1 (0.58) AKT1IKBKBCHUKNUDT1NEK1
SCHEMBL12346430 0.86 AKT1 (0.61) AKT1IKBKBCHUKNUDT1NEK1
SCHEMBL8239427 0.85 AKT1 (0.62) AKT1IKBKBCHUKKDM4ENUDT1
SCHEMBL10125362 0.84 AKT1 (0.59) AKT1IKBKBCHUKKDM4ENPC1
SCHEMBL30649183 0.84 AKT1 (0.61) AKT1IKBKBCHUKNUDT1NEK1
SCHEMBL10125059 0.84 AKT1 (0.61) AKT1IKBKBCHUKNUDT1NEK1
SCHEMBL14493849 0.83 AKT1 (0.67) AKT1HPGDSCIT
SCHEMBL4592540 0.83 AKT1 (0.67) AKT1IKBKBCHUKNUDT1NEK1
SCHEMBL14493840 0.83 NEK1 (0.64) AKT1IKBKBCHUKNUDT1NEK1
SCHEMBL14493838 0.83 AKT1 (0.66) AKT1IKBKBCHUKHPGDSCIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881983-B1 PYRROLOPYRIDINES USEFUL AS INHIBITORS OF PROTEIN KINASE VERTEX PHARMA (US) 2012-01-11 EP disclosed