SCHEMBL10125564

SCHEMBL10125564

Nc1csc(-c2ccnc3[nH]ccc23)n1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 6/20 0.64
PRKCI P41743 5/20 0.51
IKBKB O14920 3/20 0.50
CHUK O15111 3/20 0.50
AURKB Q96GD4 2/20 0.50
ROCK1 Q13464 2/20 0.50
DAPK3 O43293 1/20 0.50
JAK2 O60674 1/20 0.50
PRKD3 O94806 1/20 0.50
MAP4K4 O95819 1/20 0.50
PAK4 O96013 1/20 0.50
CSF1R P07333 1/20 0.50
RET P07949 1/20 0.50
IGF1R P08069 1/20 0.50
FGFR1 P11362 1/20 0.50
PRKACA P17612 1/20 0.50
FLT1 P17948 1/20 0.50
LTK P29376 1/20 0.50
GRK5 P34947 1/20 0.50
KDR P35968 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14494761 0.82 NUDT1 (0.64) NUDT1PRKCIIKBKBCHUKAURKB
SCHEMBL1842617 0.78 PDPK1 (0.56) ROCK1DAPK3PRKD3MAP4K4PAK4
SCHEMBL1717982 0.77 NUDT1 (0.62) NUDT1PRKCIIKBKBCHUKAURKB
SCHEMBL1719613 0.76 NUDT1 (0.57) NUDT1PRKCIIKBKBCHUKAURKB
SCHEMBL98272 0.76 ROCK1 (0.62) NUDT1PRKCIIKBKBCHUKAURKB
SCHEMBL2240671 0.76 AURKB (0.71) NUDT1PRKCIIKBKBCHUKAURKB
SCHEMBL1719341 0.76 PRKCI (0.63) NUDT1PRKCIIKBKBCHUKAURKB
SCHEMBL22160800 0.75 BRAF (0.57) NUDT1PRKCIIKBKBCHUKAURKB
SCHEMBL2239087 0.75 IKBKB (0.61) NUDT1PRKCIIKBKBCHUKAURKB
SCHEMBL1838740 0.75 CDK5 (0.64) NUDT1PRKCIIKBKBCHUKAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881983-B1 PYRROLOPYRIDINES USEFUL AS INHIBITORS OF PROTEIN KINASE VERTEX PHARMA (US) 2012-01-11 EP disclosed