SCHEMBL10129259

SCHEMBL10129259

CC(C)c1nc(N(C)C)nc(-c2ccc(F)cc2)c1/C=C/C=O

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 5/20 0.48
ALDH1A1 P00352 1/20 0.48
CYP3A4 P08684 1/20 0.48
PDE6D O43924 1/20 0.48
NR1I2 O75469 1/20 0.48
PDE4D Q08499 1/20 0.48
ABCC3 O15438 1/20 0.47
ABCC4 O15439 1/20 0.47
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17965454 0.90 HMGCR (0.46) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL17965453 0.90 HMGCR (0.46) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL697201 0.89 HMGCR (0.62) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL697202 0.89 HMGCR (0.62) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL10129258 0.87 HMGCR (0.47) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL10129222 0.86 HMGCR (0.48) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL10129521 0.82 HMGCR (0.48) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL10129470 0.82 HMGCR (0.50) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL17875116 0.81 ADORA1 (0.41) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL10433924 0.80 HMGCR (0.57) HMGCRALDH1A1CYP3A4PDE6DNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012013325-A1 PROCESS FOR THE PREPARATION OF KEY INTERMEDIATES FOR THE SYNTHESIS OF STATINS OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF LEK PHARMACEUTICALS D.D. (SI) 2012-02-02 WO disclosed