SCHEMBL1013303

SCHEMBL1013303

CC(CF)(CF)c1cc(NC(=O)O)on1

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
CNR2 P34972 10/20 0.45
CNR1 P21554 5/20 0.44
MAPK14 Q16539 5/20 0.44
RAF1 P04049 2/20 0.43
BRAF P15056 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9958632 0.88 ALDH1A1 (0.50) ALDH1A1CNR2CNR1MAPK14
SCHEMBL2635371 0.82 ALDH1A1 (0.71) ALDH1A1CNR2CNR1MAPK14RAF1
SCHEMBL1013308 0.81 RAF1 (0.47) ALDH1A1MAPK14RAF1BRAF
SCHEMBL9958104 0.80 CNR2 (0.58) ALDH1A1CNR2CNR1MAPK14
SCHEMBL1698936 0.74 EGFR (0.50) MAPK14RAF1BRAFSMN1; SMN2
SCHEMBL26789822 0.72 ALDH1A1 (0.53) ALDH1A1CNR2CNR1MAPK14SMN1; SMN2
SCHEMBL25793081 0.71 ALDH1A1 (0.55) ALDH1A1CNR2CNR1MAPK14SMN1; SMN2
SCHEMBL1896996 0.71 ALDH1A1 (0.66) ALDH1A1SMN1; SMN2
SCHEMBL25288005 0.70 ALDH1A1 (0.47) ALDH1A1MAPK14SMN1; SMN2
SCHEMBL9893018 0.69 ALDH1A1 (0.71) ALDH1A1CNR2CNR1MAPK14RAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268623-A1 QUINAZOLINE DERIVATIVES AS RAF KINASE MODULATORS AND METHODS OF USE THEREOF Ambit Biosciences Corporation (US) 2011-01-05 EP disclosed
WO-2009117080-A1 QUINAZOLINE DERIVATIVES AS RAF KINASE MODULATORS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATON (US) 2009-09-24 WO disclosed