SCHEMBL10134548

SCHEMBL10134548

CON(C)C(=O)[C@@H]1C[C@@H](C)CN1C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
UCHL1 P09936 1/20 0.39
CHRM2 P08172 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37
CYP1A2 P05177 1/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C19 P33261 1/20 0.37
NR1H2 P55055 1/20 0.35
HSD17B10 Q99714 1/20 0.33
HSD11B1 P28845 2/20 0.32
HTRA1 Q92743 1/20 0.31
PEPD P12955 1/20 0.31
GPR119 Q8TDV5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18589415 1.00 UCHL1 (0.39) UCHL1CHRM2CHRM1CHRM3CYP1A2
SCHEMBL6121364 1.00 UCHL1 (0.39) UCHL1CHRM2CHRM1CHRM3CYP1A2
SCHEMBL6121361 1.00 UCHL1 (0.39) UCHL1CHRM2CHRM1CHRM3CYP1A2
SCHEMBL18589489 1.00 UCHL1 (0.39) UCHL1CHRM2CHRM1CHRM3CYP1A2
SCHEMBL25177825 0.89 CYP1A2 (0.46) UCHL1CHRM2CHRM1CHRM3CYP1A2
SCHEMBL8135313 0.89 CYP1A2 (0.46) UCHL1CHRM2CHRM1CHRM3CYP1A2
SCHEMBL31340622 0.89 CYP1A2 (0.46) UCHL1CHRM2CHRM1CHRM3CYP1A2
SCHEMBL13086072 0.89 CYP1A2 (0.46) UCHL1CHRM2CHRM1CHRM3CYP1A2
SCHEMBL4305123 0.89 CYP1A2 (0.46) UCHL1CHRM2CHRM1CHRM3CYP1A2
SCHEMBL27393745 0.89 CYP1A2 (0.46) UCHL1CHRM2CHRM1CHRM3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12612414-B2 Nitrile SUMO inhibitors and uses thereof CIT THERAPEUTICS, INC. (US) 2026-04-28 US disclosed
US-20240360148-A1 NITRILE SUMO INHIBITORS AND USES THEREOF CIT THERAPEUTICS LLC 2024-10-31 US disclosed
EP-4373825-A1 NITRILE SUMO INHIBITORS AND USES THEREOF Suvalent Therapeutics, Inc. (US) 2024-05-29 EP disclosed
WO-2023004376-A1 NITRILE SUMO INHIBITORS AND USES THEREOF Suvalent Therapeutics, Inc. (US) 2023-01-26 WO disclosed
EP-2374794-B1 CYCLIC AMINE COMPOUNDS DAIICHI SANKYO CO LTD (JP) 2015-11-04 EP disclosed
US-20120309811-A1 P-GLYCOPROTEIN-SPECIFIC NON-COMPETITIVE PEPTIDE AND PEPTIDOMIMETIC MODULATORS UNIVERSITE CLAUDE BERNARD - LYON 1 (FR) 2012-12-06 US disclosed
US-8173631-B2 Cyclic amine compounds DAIICHI SANKYO COMPANY, LIMITED (JP) 2012-05-08 US disclosed
US-8173631-B2 Cyclic amine compounds DAIICHI SANKYO COMPANY, LIMITED (JP) 2012-05-08 US disclosed
US-20110319468-A1 CYCLIC AMINE COMPOUNDS DAIICHI SANKYO COMPANY, LIMITED (JP) 2011-12-29 US disclosed
US-20110319468-A1 CYCLIC AMINE COMPOUNDS DAIICHI SANKYO COMPANY, LIMITED (JP) 2011-12-29 US disclosed
EP-2374794-A1 CYCLIC AMINE COMPOUNDS Daiichi Sankyo Company, Limited (JP) 2011-10-12 EP disclosed
WO-2010074088-A1 CYCLIC AMINE COMPOUNDS 第一三共株式会社 (JP) 2010-07-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240360148-A1 NITRILE SUMO INHIBITORS AND USES THEREOF SUMO1, SUMO3, SUMO2 UCHL1 36/4885CHRM2 3910/4885CHRM1 2607/4885
US-12612414-B2 Nitrile SUMO inhibitors and uses thereof SUMO1, SUMO3, PSMB6 UCHL1 60/4885CHRM2 3237/4885CHRM1 2156/4885
US-20120309811-A1 P-GLYCOPROTEIN-SPECIFIC NON-COMPETITIVE PEPTIDE AND PEPTIDOMIMETIC MODULATORS ABCB1, ABCG2, SELPLG UCHL1 4707/4885CHRM2 4700/4885CHRM1 4319/4885
US-20110319468-A1 CYCLIC AMINE COMPOUNDS RYR2, CASR, RYR1 UCHL1 4548/4885CHRM2 252/4885CHRM1 232/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.