SCHEMBL10134802

SCHEMBL10134802

COc1ccccc1NC(=O)c1cncc(Nc2ccccc2)n1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.54
AHR P35869 2/20 0.54
MEN1 O00255 2/20 0.54
BRAF P15056 4/20 0.53
MAPT P10636 2/20 0.51
P4HTM Q9NXG6 1/20 0.51
STAT3 P40763 1/20 0.50
STAT1 P42224 1/20 0.50
IRAK4 Q9NWZ3 1/20 0.49
KDM4E B2RXH2 1/20 0.49
NPC1 O15118 1/20 0.48
ALDH1A1 P00352 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
CDK2 P24941 1/20 0.48
HTT P42858 1/20 0.47
CD38 P28907 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10134797 0.82 CDK2 (0.57) BRAFKDM4ENPC1ALDH1A1SMN1; SMN2
SCHEMBL10134867 0.79 RAB9A (0.58) KMT2AAHRMEN1BRAFMAPT
SCHEMBL560178 0.78 ATR (0.63) KMT2AAHRMEN1MAPTP4HTM
SCHEMBL10134816 0.77 JAK2 (0.53) KMT2ABRAFSTAT3KDM4ENPC1
SCHEMBL10134810 0.74 RAB9A (0.56) KMT2AMEN1IRAK4KDM4ENPC1
SCHEMBL23413101 0.73 MEN1 (0.54) KMT2AMEN1BRAFMAPTSTAT3
SCHEMBL29887175 0.73 MEN1 (0.54) KMT2AMEN1BRAFMAPTSTAT3
SCHEMBL23413488 0.72 MAPT (0.55) KMT2AMEN1BRAFMAPTSTAT3
SCHEMBL23413150 0.72 MAPT (0.53) KMT2AMEN1BRAFMAPTSTAT3
SCHEMBL23413089 0.72 MEN1 (0.55) KMT2AAHRMEN1BRAFMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8962631-B2 Compounds useful as inhibitors of ATR kinase VERTEX PHARMACEUTICALS INCORPORATED (US) 2015-02-24 US disclosed
US-20120035407-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-02-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120035407-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE ATR, CHEK1, CHEK2 KMT2A 1532/4885AHR 2654/4885MEN1 2408/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.