SCHEMBL10146007

SCHEMBL10146007

Cn1c(=O)n(CC2CCCC2)c2ccc(-c3cc(Oc4ccnc(N)c4)ccc3C#N)cc21

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 2/20 0.43
PARG Q86W56 4/20 0.38
XDH P47989 1/20 0.35
KDM1A O60341 1/20 0.35
RAF1 P04049 1/20 0.34
BRAF P15056 1/20 0.34
PIK3CA P42336 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
SCN9A Q15858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14992645 0.92 GRM2 (0.44) GRM2PARGXDHKDM1ARAF1
SCHEMBL627802 0.90 GRM2 (0.46) GRM2PARGXDHKDM1ARAF1
SCHEMBL627819 0.88 GRM2 (0.44) GRM2PARGXDHPIK3CAGRIN1
SCHEMBL626150 0.85 PIK3CA (0.41) GRM2XDHPIK3CA
SCHEMBL10145839 0.82 PIK3CA (0.44) GRM2PARGPIK3CAGRIN1GRIN2B
SCHEMBL10146006 0.80 PARG (0.40) GRM2PARGPIK3CAGRIN1GRIN2B
SCHEMBL14992707 0.78 PARG (0.47) GRM2PARG
SCHEMBL627523 0.77 PARG (0.45) GRM2PARGXDHKDM1A
SCHEMBL14992922 0.76 GRM2 (0.40) GRM2PARGXDH
SCHEMBL627295 0.76 GRM2 (0.43) GRM2PARGGRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021382-A1 POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 MERCK SHARP & DOHME CORP. (US) 2012-02-16 WO disclosed