SCHEMBL10146348

SCHEMBL10146348

Cn1c(=O)n(CC2CC2)c2ccc(-c3cccc(Oc4ccccc4N)c3)cc21

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.43
PARG Q86W56 4/20 0.41
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
ICMT O60725 2/20 0.37
BACE1 P56817 1/20 0.36
CRHR1 P34998 3/20 0.36
CRHR2 Q13324 1/20 0.36
GRIN1 Q05586 4/20 0.36
GRIN2B Q13224 4/20 0.36
TRIM24 O15164 2/20 0.35
BRD4 O60885 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10145942 0.88 NPC1 (0.43) GRM2PARGALDH1A1ICMTCRHR1
SCHEMBL625527 0.88 GRM2 (0.51) GRM2PARGICMTCRHR1CRHR2
SCHEMBL10146339 0.87 PARG (0.43) GRM2PARGALDH1A1ICMTBACE1
SCHEMBL10146345 0.86 PARG (0.42) GRM2PARGALDH1A1GAAICMT
SCHEMBL14992323 0.86 GRM2 (0.41) GRM2PARGGAAICMTCRHR1
SCHEMBL10146010 0.85 PARG (0.39) GRM2PARGICMTBACE1CRHR1
SCHEMBL10146338 0.83 GRIN1 (0.48) GRM2PARGICMTCRHR1CRHR2
SCHEMBL10146006 0.83 PARG (0.40) GRM2PARGICMTBACE1CRHR1
SCHEMBL10145997 0.82 PARG (0.42) GRM2PARGICMTCRHR1CRHR2
SCHEMBL625690 0.82 GRM2 (0.43) GRM2PARGICMTCRHR1CRHR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021382-A1 POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 MERCK SHARP & DOHME CORP. (US) 2012-02-16 WO disclosed