SCHEMBL10146398

SCHEMBL10146398

CCc1cc2nc(C)[nH]c2cc1Cl

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.53
HTT P42858 2/20 0.53
GRIN2D O15399 2/20 0.51
GRIN3B O60391 2/20 0.51
GRIN1 Q05586 2/20 0.51
GRIN2A Q12879 2/20 0.51
GRIN2B Q13224 2/20 0.51
GRIN2C Q14957 2/20 0.51
GRIN3A Q8TCU5 2/20 0.51
ALDH1A1 P00352 2/20 0.50
POLB P06746 2/20 0.42
HPGD P15428 2/20 0.42
MAPT P10636 2/20 0.42
KDM4E B2RXH2 1/20 0.42
PARP1 P09874 1/20 0.41
HSP90AA1 P07900 1/20 0.41
ESR2 Q92731 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CHRNB2 P17787 1/20 0.40
CHRNA4 P43681 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL316047 0.81 ALDH1A1 (0.60) GAAHTTGRIN2DGRIN3BGRIN1
SCHEMBL10292838 0.79 MAPT (0.46) GAAHTTALDH1A1POLBHPGD
SCHEMBL12020717 0.78 ALDH1A1 (0.56) GAAHTTGRIN2DGRIN3BGRIN1
SCHEMBL24463172 0.75 ALDH1A1 (0.53) GAAHTTALDH1A1POLBHPGD
SCHEMBL8265257 0.75 ALDH1A1 (0.53) GAAHTTALDH1A1POLBHPGD
SCHEMBL29954905 0.75 ALDH1A1 (0.53) GAAHTTALDH1A1POLBHPGD
SCHEMBL5752586 0.75 ALDH1A1 (0.53) GAAHTTALDH1A1POLBHPGD
SCHEMBL13041691 0.74 ALDH1A1 (0.59) GAAHTTALDH1A1POLBHPGD
SCHEMBL8264566 0.74 ALDH1A1 (0.56) GAAHTTGRIN2DGRIN3BGRIN1
SCHEMBL14496860 0.73 MAPT (0.46) GAAHTTALDH1A1POLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012009217-A1 SPIROCYCLIC COMPOUNDS MERCK SHARP & DOHME CORP. (US) 2012-01-19 WO disclosed