SCHEMBL10147083

SCHEMBL10147083

O=C(O)CC1CCC2(CC1)CCN(c1ccc(-c3nc4cnccc4[nH]3)cn1)CC2

nearest known ligand 0.70

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 19/20 0.70
KCNH2 Q12809 17/20 0.70
CYP2C9 P11712 4/20 0.70
CYP3A4 P08684 2/20 0.70
ADORA2A P29274 5/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10146410 0.89 DGAT1 (0.76) DGAT1KCNH2CYP2C9CYP3A4ADORA2A
SCHEMBL10146483 0.85 DGAT1 (0.81) DGAT1KCNH2CYP2C9CYP3A4ADORA2A
SCHEMBL10146540 0.85 DGAT1 (0.79) DGAT1KCNH2CYP2C9CYP3A4ADORA2A
SCHEMBL10146477 0.84 DGAT1 (0.80) DGAT1KCNH2CYP2C9CYP3A4ADORA2A
SCHEMBL10147076 0.84 DGAT1 (0.65) DGAT1KCNH2CYP2C9CYP3A4ADORA2A
SCHEMBL10146413 0.84 DGAT1 (0.88) DGAT1KCNH2CYP2C9CYP3A4ADORA2A
SCHEMBL10147230 0.81 DGAT1 (0.66) DGAT1KCNH2CYP2C9CYP3A4ADORA2A
SCHEMBL10147078 0.81 DGAT1 (0.78) DGAT1KCNH2CYP2C9CYP3A4ADORA2A
SCHEMBL10147222 0.81 DGAT1 (0.64) DGAT1KCNH2CYP2C9CYP3A4ADORA2A
SCHEMBL10146466 0.81 DGAT1 (0.65) DGAT1KCNH2CYP2C9CYP3A4ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012009217-A1 SPIROCYCLIC COMPOUNDS MERCK SHARP & DOHME CORP. (US) 2012-01-19 WO disclosed