SCHEMBL10147484

SCHEMBL10147484

CN1CC(C2=C(c3cccs3)C(c3cc(O)c(C(=O)O)c(F)c3)CC(=O)N2)C=N1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 1/20 0.32
FEN1 P39748 1/20 0.32
ERCC4 Q92889 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
MAPK1 P28482 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL368840 0.68 ALDH1A1 (0.37) KMT2AALDH1A1MAPTMAPK1L3MBTL1
SCHEMBL367874 0.66 TP53 (0.31) ALDH1A1
SCHEMBL367884 0.61 KDM4E (0.39) KMT2AALDH1A1MAPTMAPK1L3MBTL1
SCHEMBL19328808 0.56 ERN1 (0.55) MEN1KMT2AMAPTL3MBTL1
SCHEMBL873514 0.55 KDM4E (0.50) MEN1KMT2AALDH1A1MAPTL3MBTL1
SCHEMBL2721939 0.52 ALDH1A1 (0.55) MEN1KMT2AALDH1A1MAPTMAPK1
SCHEMBL11642810 0.51 ALDH1A1 (0.44) ERCC1FEN1ERCC4MEN1KMT2A
SCHEMBL7489462 0.51 EGFR (0.52) MEN1KMT2AALDH1A1MAPTMAPK1
SCHEMBL27577897 0.51 ERCC1 (0.44) ERCC1FEN1ERCC4MEN1KMT2A
SCHEMBL20773225 0.50 MAPT (0.45) MEN1KMT2AALDH1A1MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012009227-A1 NOVEL DIHYDROPYRIDIN-2(1H)-ONE COMPOUNDS AS S-NITROSOGLUTATHIONE REDUCTASE INHIBITORS AND NEUROKININ-3 RECEPTOR ANTAGONISTS N30 PHARMACEUTICALS, LLC (US) 2012-01-19 WO disclosed