SCHEMBL10153606

SCHEMBL10153606

CC(C)(C)NC(=O)C1C(=O)N(O)C(=O)c2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 11/20 0.48
KCNH2 Q12809 5/20 0.48
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
NCOR2 Q9Y618 1/20 0.41
PKM P14618 1/20 0.40
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31653994 1.00 KCNA5 (0.48) KCNA5KCNH2HDAC3HDAC4HDAC7
SCHEMBL19380274 0.84 HDAC4 (0.44) KCNA5KCNH2HDAC3HDAC4HDAC7
SCHEMBL9958705 0.82 HDAC4 (0.62) HDAC3HDAC4HDAC7HDAC8HDAC6
SCHEMBL10153609 0.82 MEN1 (0.47) HDAC3HDAC4HDAC7HDAC8HDAC6
SCHEMBL31653962 0.82 MEN1 (0.47) HDAC3HDAC4HDAC7HDAC8HDAC6
SCHEMBL10154010 0.81 MAPT (0.44) KCNA5HDAC3HDAC4HDAC7HDAC8
SCHEMBL22461359 0.80 HDAC4 (0.61) KCNA5KCNH2HDAC3HDAC4HDAC7
SCHEMBL10153604 0.78 KCNA5 (0.47) KCNA5KCNH2HDAC3HDAC4HDAC7
SCHEMBL19380301 0.78 HDAC3 (0.40) HDAC3HDAC4HDAC7HDAC8HDAC6
SCHEMBL9958675 0.77 KMT2A (0.50) KCNA5KCNH2MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed