SCHEMBL10153701

SCHEMBL10153701

CCOC(=O)CNC(=O)C1C(=O)N(O)C(=O)c2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.57
ALDH1A1 P00352 6/20 0.52
NPSR1 Q6W5P4 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.46
CYP1A2 P05177 1/20 0.42
PPID Q08752 1/20 0.41
USP2 O75604 2/20 0.39
KDM4E B2RXH2 2/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CA12 O43570 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
PIN1 Q13526 1/20 0.39
PIN4 Q9Y237 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
IDO1 P14902 1/20 0.38
LTA4H P09960 1/20 0.38
MMP2 P08253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10153971 0.82 POLB (0.50) POLBALDH1A1NPSR1SMN1; SMN2CYP1A2
SCHEMBL10153604 0.82 KCNA5 (0.47) POLBALDH1A1NPSR1SMN1; SMN2MEN1
SCHEMBL10153314 0.80 KMT2A (0.54) ALDH1A1NPSR1SMN1; SMN2KDM4EMEN1
SCHEMBL10153707 0.79 KMT2A (0.55) ALDH1A1NPSR1SMN1; SMN2KDM4EMEN1
SCHEMBL9952669 0.78 KMT2A (0.54) ALDH1A1NPSR1SMN1; SMN2KDM4EMEN1
SCHEMBL10153662 0.78 KMT2A (0.54) ALDH1A1NPSR1SMN1; SMN2KDM4EMEN1
SCHEMBL9959705 0.78 KMT2A (0.54) ALDH1A1NPSR1SMN1; SMN2KDM4EMEN1
SCHEMBL9959242 0.78 KMT2A (0.54) ALDH1A1NPSR1SMN1; SMN2KDM4EMEN1
SCHEMBL9952553 0.78 KMT2A (0.54) ALDH1A1NPSR1SMN1; SMN2KDM4EMEN1
SCHEMBL10154090 0.78 KCNA5 (0.47) ALDH1A1SMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed