SCHEMBL10153707

SCHEMBL10153707

CCCCCNC(=O)C1C(=O)N(O)C(=O)c2ccccc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.55
MEN1 O00255 2/20 0.55
ASAH1 Q13510 1/20 0.51
MAPT P10636 1/20 0.50
GSK3B P49841 1/20 0.47
KCNA5 P22460 4/20 0.46
KCNH2 Q12809 1/20 0.46
ALDH1A1 P00352 3/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
KDM4E B2RXH2 1/20 0.45
NLRP3 Q96P20 1/20 0.45
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
DRD3 P35462 1/20 0.43
GAA P10253 1/20 0.42
NAAA Q02083 1/20 0.41
NPC1 O15118 1/20 0.40
ALOX15 P16050 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9959242 0.99 KMT2A (0.54) KMT2AMEN1ASAH1MAPTGSK3B
SCHEMBL10153662 0.99 KMT2A (0.54) KMT2AMEN1ASAH1MAPTGSK3B
SCHEMBL9952669 0.99 KMT2A (0.54) KMT2AMEN1ASAH1MAPTGSK3B
SCHEMBL9959705 0.99 KMT2A (0.54) KMT2AMEN1ASAH1MAPTGSK3B
SCHEMBL9952553 0.99 KMT2A (0.54) KMT2AMEN1ASAH1MAPTGSK3B
SCHEMBL10153314 0.96 KMT2A (0.54) KMT2AMEN1ASAH1MAPTGSK3B
SCHEMBL10153604 0.91 KCNA5 (0.47) KMT2AMEN1ASAH1MAPTKCNA5
SCHEMBL9958620 0.86 DRD2 (0.44) KMT2AMEN1MAPTKCNA5KCNH2
SCHEMBL10154063 0.80 KMT2A (0.47) KMT2AMEN1ASAH1MAPTGSK3B
SCHEMBL9959738 0.80 KMT2A (0.47) KMT2AMEN1ASAH1MAPTGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed