SCHEMBL10154458

SCHEMBL10154458

CCCCC(N)c1ccc(C(=O)OC)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.53
ERAP2 Q6P179 2/20 0.52
LNPEP Q9UIQ6 2/20 0.52
MAPT P10636 2/20 0.49
NPC1 O15118 1/20 0.48
CASP1 P29466 1/20 0.48
RAB9A P51151 1/20 0.48
LOXL2 Q9Y4K0 1/20 0.47
SLC2A1 P11166 1/20 0.47
HPGD P15428 1/20 0.46
MGLL Q99685 1/20 0.46
SLC6A2 P23975 1/20 0.45
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
CA12 O43570 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12328884 1.00 DPP4 (0.53) DPP4ERAP2LNPEPMAPTNPC1
SCHEMBL12326257 0.95 SLC2A1 (0.52) DPP4ERAP2LNPEPMAPTNPC1
SCHEMBL14551497 0.95 SLC2A1 (0.52) DPP4ERAP2LNPEPMAPTNPC1
SCHEMBL20874440 0.91 DPP4 (0.49) DPP4ERAP2LNPEPMAPTNPC1
SCHEMBL12326223 0.90 DPP4 (0.56) DPP4ERAP2LNPEPMAPTNPC1
SCHEMBL14550338 0.90 DPP4 (0.56) DPP4ERAP2LNPEPMAPTNPC1
SCHEMBL14550548 0.85 CA12 (0.50) DPP4ERAP2LNPEPMAPTNPC1
SCHEMBL14551239 0.84 DPP4 (0.56) DPP4MAPTNPC1RAB9ALOXL2
SCHEMBL12326121 0.84 DPP4 (0.56) DPP4MAPTNPC1RAB9ALOXL2
SCHEMBL1765662 0.84 NPC1 (0.50) ERAP2LNPEPMAPTNPC1CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012009226-A1 SUBSTITUTED IMIDAZOLONES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE MERCK SHARP & DOHME CORP. (US) 2012-01-19 WO disclosed
WO-2011119559-A1 NOVEL SPIRO IMIDAZOLONES AS GLUCAGON RECEPTOR ANTAGONISTS, COMPOSITIONS, AND METHODS FOR THEIR USE SCHERING CORPORATION (US) 2011-09-29 WO disclosed