SCHEMBL10154672

SCHEMBL10154672

CNC(=O)OC1CN(C)C1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 4/20 0.44
CHRM3 P20309 5/20 0.43
CHRM4 P08173 4/20 0.43
SMN1; SMN2 Q16637 1/20 0.35
ATM Q13315 1/20 0.34
EPHX1 P07099 2/20 0.33
BCHE P06276 2/20 0.33
CHRM5 P08912 3/20 0.33
CHRM2 P08172 2/20 0.31
CYP2D6 P10635 1/20 0.30
POLB P06746 1/20 0.30
HTT P42858 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29680526 0.84 CHRM1 (0.49) CHRM1CHRM3CHRM4SMN1; SMN2CHRM5
SCHEMBL14852963 0.81 CHRM1 (0.43) CHRM1ATMEPHX1BCHE
SCHEMBL18587782 0.81 CHRM3 (0.42) CHRM1CHRM3CHRM4SMN1; SMN2ATM
SCHEMBL30916849 0.79 CHRM3 (0.49) CHRM1CHRM3CHRM4SMN1; SMN2ATM
SCHEMBL17082702 0.79 CHRM1 (0.42) CHRM1SMN1; SMN2ATMEPHX1BCHE
SCHEMBL25595757 0.78 CHRM4 (0.40) CHRM3CHRM4SMN1; SMN2ATMBCHE
SCHEMBL14299898 0.78 CHRM1 (0.41) CHRM1CHRM3CHRM4ATMEPHX1
SCHEMBL11929075 0.78 CHRM1 (0.41) CHRM1ATMEPHX1BCHE
SCHEMBL10150974 0.78 CHRM4 (0.40) CHRM3CHRM4SMN1; SMN2EPHX1CYP2D6
SCHEMBL103736 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023107714-A2 METHODS FOR TREATING NEUROLOGICAL DISORDERS PROTHENA BIOSCIENCES LIMITED (IE) 2023-06-15 WO disclosed
WO-2023081312-A1 SMALL MOLECULE INDUCERS OF AUTOPHAGY Vir Biotechnology, Inc. (US) 2023-05-11 WO disclosed
US-9765087-B2 Benzimidazole derivatives ENANTA PHARMACEUTICALS, INC. (US) 2017-09-19 US disclosed
US-20170114046-A1 NOVEL BENZIMIDAZOLE DERIVATIVES ENANTA PHARM INC (US) 2017-04-27 US disclosed
US-20140341851-A1 NOVEL BENZIMIDAZOLE DERIVATIVES ENANTA PHARMACEUTICALS, INC. (US) 2014-11-20 US disclosed
US-20140193363-A1 NOVEL BENZIMIDAZOLE DERIVATIVES ENANTA PHARMACEUTICALS, INC. (US) 2014-07-10 US disclosed
US-8673954-B2 Benzimidazole derivatives ENANTA PHARMACEUTICALS, INC. (US) 2014-03-18 US disclosed
US-8507522-B2 Hepatitis C virus inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2013-08-13 US disclosed
US-8242156-B2 Linked dibenzimidazole derivatives ENANTA PHARMACEUTICALS, INC. (US) 2012-08-14 US disclosed
US-8101643-B2 Benzimidazole derivatives ENANTA PHARMACEUTICALS, INC. (US) 2012-01-24 US disclosed
US-20100260715-A1 HEPATITIS C VIRUS INHIBITORS ENANTA PHARMACEUTICALS, INC. 2010-10-14 US disclosed
US-20100233122-A1 NOVEL BENZIMIDAZOLE DERIVATIVES ENANTA PHARMACEUTICALS, INC. 2010-09-16 US disclosed
US-20100221215-A1 LINKED DIBENZIMIDAZOLE DERIVATIVES ENANTA PHARMACEUTICALS, INC. 2010-09-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170114046-A1 NOVEL BENZIMIDAZOLE DERIVATIVES EIF2AK2, ZC3HAV1, HAVCR2 CHRM1 4784/4885CHRM3 4599/4885CHRM4 4809/4885
US-20100260715-A1 HEPATITIS C VIRUS INHIBITORS HAVCR2, SLC10A1, EIF2AK2 CHRM1 4800/4885CHRM3 4574/4885CHRM4 4823/4885
US-20100233122-A1 NOVEL BENZIMIDAZOLE DERIVATIVES EIF2AK2, ZC3HAV1, HAVCR2 CHRM1 4784/4885CHRM3 4599/4885CHRM4 4809/4885
US-20100221215-A1 LINKED DIBENZIMIDAZOLE DERIVATIVES EIF2AK2, NSUN2, ZC3HAV1 CHRM1 4857/4885CHRM3 4759/4885CHRM4 4859/4885
US-20140193363-A1 NOVEL BENZIMIDAZOLE DERIVATIVES EIF2AK2, ZC3HAV1, HAVCR2 CHRM1 4784/4885CHRM3 4599/4885CHRM4 4809/4885
US-20140341851-A1 NOVEL BENZIMIDAZOLE DERIVATIVES EIF2AK2, ZC3HAV1, HAVCR2 CHRM1 4784/4885CHRM3 4599/4885CHRM4 4809/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.