SCHEMBL10156528

SCHEMBL10156528

CCc1nc(C(N)=O)c(Nc2ccc(CN3CCN(C)CC3)cc2C)nc1C

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EML4 Q9HC35 10/20 0.44
ALK Q9UM73 10/20 0.44
CCR5 P51681 1/20 0.43
IKBKE Q14164 5/20 0.43
TBK1 Q9UHD2 4/20 0.43
ENPP2 Q13822 2/20 0.42
RET P07949 3/20 0.41
ROS1 P08922 3/20 0.41
FLT3 P36888 3/20 0.41
TNIK Q9UKE5 1/20 0.41
GRM2 Q14416 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL328289 0.91 IKBKE (0.44) EML4ALKCCR5IKBKETBK1
SCHEMBL10129612 0.84 EML4 (0.65) EML4ALKRETROS1FLT3
SCHEMBL17690612 0.82 EML4 (0.47) EML4ALKRETROS1FLT3
SCHEMBL17689742 0.80 PARP1 (0.40) EML4ALKIKBKETBK1FLT3
SCHEMBL10157702 0.79 EML4 (0.54) EML4ALKRETROS1FLT3
SCHEMBL10126816 0.76 IKBKE (0.55) EML4ALKIKBKETBK1RET
SCHEMBL16206813 0.75 EML4 (0.51) EML4ALKRETROS1FLT3
SCHEMBL10155938 0.74 PLAU (0.38) EML4ALK
SCHEMBL16206819 0.72 ALK (0.47) EML4ALKRETROS1FLT3
SCHEMBL16195799 0.72 EGFR (0.61) EML4ALKIKBKETBK1RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120040968-A1 DIAMINO HETEROCYCLIC CARBOXAMIDE COMPOUND WATERS TECHNOLOGIES CORPORATION (US) 2012-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120040968-A1 DIAMINO HETEROCYCLIC CARBOXAMIDE COMPOUND EML4, ALK, ERBB4 EML4 1/4885ALK 2/4885CCR5 2406/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.