SCHEMBL10157693

SCHEMBL10157693

COC(=O)CCNc1cc(C(C)(C)C)nc(Cl)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
PGK1 P00558 1/20 0.37
CA1 P00915 4/20 0.37
CA2 P00918 4/20 0.37
CA12 O43570 3/20 0.37
CA9 Q16790 3/20 0.37
CA14 Q9ULX7 3/20 0.37
HRH4 Q9H3N8 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ESR1 P03372 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
KAT2B Q92831 1/20 0.33
EGFR P00533 1/20 0.32
CA3 P07451 1/20 0.32
CA4 P22748 1/20 0.32
CA6 P23280 1/20 0.32
CA5A P35218 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10157581 0.88 SMN1; SMN2 (0.41) KMT2AMEN1ALDH1A1POLBPGK1
SCHEMBL19072323 0.78 LMNA (0.50) KMT2AMEN1ALDH1A1POLBPGK1
SCHEMBL10157584 0.75 KDM6A (0.52) KMT2AALDH1A1
SCHEMBL11292565 0.70 PTGDR (0.41) KMT2AMEN1ALDH1A1POLBPGK1
SCHEMBL3418234 0.68 LMNA (0.45) KMT2AHRH4SMN1; SMN2ESR1MAPT
SCHEMBL10266953 0.68 CYP2D6 (0.41) KMT2AMEN1ALDH1A1CA1CA2
SCHEMBL5063085 0.66 PRNP (0.44) ALDH1A1CA12CA9CA14HRH4
SCHEMBL12257760 0.66 HRH4 (0.53) KMT2AMEN1ALDH1A1HRH4SMN1; SMN2
SCHEMBL12615675 0.66 CYP2D6 (0.56) KMT2AALDH1A1POLBHRH4SMN1; SMN2
SCHEMBL19072212 0.66 KMT2A (0.41) KMT2AMEN1ALDH1A1POLBCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012052390-A1 N-2-(2-PYRIDINYL)-4-PYRIMIDINYL-BETA-ALANINE DERIVATIVES AS INHIBITORS OF HISTONE DEMETHYLASE JMJD3 GLAXO GROUP LIMITED (GB) 2012-04-26 WO disclosed