SCHEMBL1015823

SCHEMBL1015823

NC(=O)c1ccc(C(=O)Nc2ccc(Cl)c(-c3ccccn3)c2)cc1

nearest known ligand 0.84

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALB P02768 1/20 0.58
HTR1A P08908 1/20 0.58
SLC6A2 P23975 1/20 0.58
PDE4A P27815 1/20 0.58
OPRM1 P35372 1/20 0.58
DRD3 P35462 1/20 0.58
HTR2B P41595 1/20 0.58
SLC6A3 Q01959 1/20 0.58
PDE4D Q08499 1/20 0.58
SHH Q15465 1/20 0.58
USP28 Q96RU2 1/20 0.58
SLC29A1 Q99808 1/20 0.58
SMO Q99835 1/20 0.58
ABCG2 Q9UNQ0 1/20 0.58
GRM4 Q14833 2/20 0.54
BCAT2 O15382 1/20 0.53
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
KCNK3 O14649 1/20 0.51
KCNK9 Q9NPC2 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28386672 0.91 ALB (0.64) ALBHTR1ASLC6A2PDE4AOPRM1
SCHEMBL1015524 0.91 ALB (0.58) ALBHTR1ASLC6A2PDE4AOPRM1
SCHEMBL1017617 0.90 ALB (0.55) ALBHTR1ASLC6A2PDE4AOPRM1
SCHEMBL15424139 0.89 ALB (0.59) ALBHTR1ASLC6A2PDE4AOPRM1
SCHEMBL1017518 0.89 ALB (0.59) ALBHTR1ASLC6A2PDE4AOPRM1
SCHEMBL1018176 0.89 USP28 (0.68) ALBHTR1ASLC6A2PDE4AOPRM1
SCHEMBL30572237 0.89 USP28 (0.68) ALBHTR1ASLC6A2PDE4AOPRM1
SCHEMBL17783734 0.88 NPC1 (0.59) ALBHTR1ASLC6A2PDE4AOPRM1
SCHEMBL1017948 0.87 USP28 (0.55) ALBHTR1ASLC6A2PDE4AOPRM1
SCHEMBL1251379 0.86 ALB (0.54) ALBHTR1ASLC6A2PDE4AOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2271642-A2 PYRIDYL INHIBITORS OF HEDGEHOG SIGNALLING Genentech, Inc. (US) 2011-01-12 EP disclosed