SCHEMBL10168628

SCHEMBL10168628

CC(C)N1CCCC2(CCN(C)C2=O)C1

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 2/20 0.32
GRIN2A Q12879 2/20 0.32
LTA4H P09960 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12832197 0.91 CYP2D6 (0.33) GRIN1GRIN2A
SCHEMBL25900548 0.86 GRIN1 (0.36) GRIN1GRIN2ALTA4H
SCHEMBL19077884 0.86 SMN1; SMN2 (0.36) GRIN1GRIN2ALTA4H
SCHEMBL22155723 0.83 ACACB (0.35)
SCHEMBL9963247 0.83 LTA4H (0.37) GRIN1GRIN2ALTA4H
SCHEMBL16559762 0.82 CYP2D6 (0.34)
SCHEMBL16559764 0.80 CYP2D6 (0.39)
SCHEMBL9963245 0.80 CYP2D6 (0.39) GRIN1GRIN2ALTA4H
SCHEMBL20420099 0.80 ACACB (0.33)
SCHEMBL10186825 0.79 GRIN1 (0.38) GRIN1GRIN2ALTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200197391-A1 COMPOUNDS THAT PARTICIPATE IN COOPERATIVE BINDING AND USES THEREOF Revolution Medicines, Inc. 2020-06-25 US disclosed
US-8586751-B2 Nicotinamide compounds useful as kinase modulators BRISTOL-MYERS SQUIBB COMPANY (US) 2013-11-19 US disclosed
US-20120082702-A1 NICOTINAMIDE COMPOUNDS USEFUL AS KINASE MODULATORS BRISTOL-MEYERS SQUIBB COMPANY 2012-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200197391-A1 COMPOUNDS THAT PARTICIPATE IN COOPERATIVE BINDING AND USES THEREOF KRAS, NRAS, HRAS GRIN1 4674/4885GRIN2A 4673/4885LTA4H 4302/4885
US-20120082702-A1 NICOTINAMIDE COMPOUNDS USEFUL AS KINASE MODULATORS NADK, BTK, NAMPT GRIN1 1342/4885GRIN2A 2444/4885LTA4H 1365/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.