SCHEMBL10175110

SCHEMBL10175110

N#Cc1ccc2nc(-c3cncc4ccccc34)n(C3CC3)c2c1

nearest known ligand 0.62

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 20/20 0.62
CYP11B1 P15538 17/20 0.62
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL428457 0.83 CYP11B2 (0.71) CYP11B2CYP11B1CYP3A4
SCHEMBL17896652 0.83 CYP11B2 (0.53) CYP11B2CYP11B1CYP3A4
SCHEMBL17896698 0.83 CYP11B2 (0.60) CYP11B2CYP11B1CYP3A4
SCHEMBL17896610 0.82 CYP11B2 (0.53) CYP11B2CYP11B1
SCHEMBL17896615 0.80 CYP11B2 (0.68) CYP11B2CYP11B1CYP3A4
SCHEMBL431913 0.80 CYP11B2 (0.67) CYP11B2CYP11B1CYP3A4
SCHEMBL31412053 0.79 CYP11B2 (0.74) CYP11B2CYP11B1
SCHEMBL20337766 0.79 CYP11B2 (0.74) CYP11B2CYP11B1
SCHEMBL17896606 0.79 CYP11B2 (0.66) CYP11B2CYP11B1
SCHEMBL17896608 0.79 CYP11B2 (0.66) CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed