SCHEMBL10175362

SCHEMBL10175362

Cc1ccncc1-c1nc2ccc(Cl)cc2n1C1CC1

nearest known ligand 0.69

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 15/20 0.69
CYP11B1 P15538 13/20 0.69
PDE10A Q9Y233 4/20 0.62
PDE2A O00408 3/20 0.62
CYP3A4 P08684 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896657 0.85 CYP11B2 (0.69) CYP11B2CYP11B1PDE10APDE2ACYP3A4
SCHEMBL10175598 0.85 CYP11B2 (0.76) CYP11B2CYP11B1PDE10ACYP3A4
SCHEMBL22791690 0.82 CYP11B1 (0.69) CYP11B2CYP11B1CYP3A4
SCHEMBL10175597 0.81 CYP11B2 (1.00) CYP11B2CYP11B1CYP3A4
SCHEMBL17896698 0.81 CYP11B2 (0.60) CYP11B2CYP11B1CYP3A4
SCHEMBL17896731 0.81 CYP11B1 (0.72) CYP11B2CYP11B1CYP3A4
SCHEMBL10175358 0.81 PDE10A (0.65) CYP11B2CYP11B1PDE10APDE2A
SCHEMBL17896695 0.79 CYP11B2 (0.55) CYP11B2CYP11B1CYP3A4
SCHEMBL10175365 0.79 CYP11B2 (1.00) CYP11B2CYP11B1
SCHEMBL20337667 0.78 CYP11B1 (0.70) CYP11B2CYP11B1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed