SCHEMBL10175422

SCHEMBL10175422

COc1ccc2nc(-c3cccnc3)n(C3CC3)c2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 19/20 1.00
CYP11B1 P15538 14/20 1.00
HTR2B P41595 1/20 0.56
HTR6 P50406 1/20 0.56
CYP17A1 P05093 1/20 0.49
CYP19A1 P11511 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL461190 0.91 CYP11B2 (0.83) CYP11B2CYP11B1HTR2BHTR6CYP17A1
SCHEMBL20337711 0.87 CYP11B2 (0.77) CYP11B2CYP11B1HTR2BCYP19A1
SCHEMBL17896585 0.85 CYP11B2 (0.76) CYP11B2CYP11B1HTR2BHTR6CYP19A1
SCHEMBL10175365 0.82 CYP11B2 (1.00) CYP11B2CYP11B1HTR2BHTR6
SCHEMBL460209 0.82 CYP11B2 (1.00) CYP11B2CYP11B1HTR2BHTR6CYP19A1
SCHEMBL17896653 0.82 CYP11B2 (0.74) CYP11B2CYP11B1HTR2BHTR6CYP19A1
SCHEMBL17896588 0.80 CYP11B2 (1.00) CYP11B2CYP11B1HTR2BHTR6
SCHEMBL10175582 0.79 CYP11B2 (1.00) CYP11B2CYP11B1HTR2BHTR6CYP19A1
SCHEMBL458680 0.79 CYP11B2 (1.00) CYP11B2CYP11B1HTR2BHTR6
SCHEMBL17896584 0.79 CYP11B2 (0.69) CYP11B2CYP11B1HTR2BHTR6CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed