SCHEMBL10176193

SCHEMBL10176193

CC(C)(O)c1cncc(C(=O)O)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 6/20 0.55
ALDH1A1 P00352 4/20 0.50
KDM4E B2RXH2 3/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
LMNA P02545 2/20 0.50
POLB P06746 1/20 0.50
DDO Q99489 1/20 0.50
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
RAF1 P04049 1/20 0.40
CYP11B2 P19099 6/20 0.39
APP P05067 1/20 0.38
GAA P10253 1/20 0.38
HCAR3 P49019 1/20 0.38
CYP11B1 P15538 3/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30236806 1.00 HCAR2 (0.55) HCAR2ALDH1A1KDM4EMEN1KMT2A
SCHEMBL12412645 0.86 HCAR2 (0.57) HCAR2ALDH1A1KDM4EMEN1KMT2A
SCHEMBL28283555 0.83 HCAR2 (0.53) HCAR2ALDH1A1KDM4EMEN1KMT2A
SCHEMBL31032251 0.83 HCAR2 (0.53) HCAR2ALDH1A1KDM4EMEN1KMT2A
SCHEMBL22778668 0.80 HCAR2 (0.50) HCAR2ALDH1A1KDM4EMEN1KMT2A
SCHEMBL431513 0.80 ATM (0.59) ALDH1A1KDM4ELMNAPOLBCYP2C9
SCHEMBL17896592 0.80 CYP11B2 (0.35) HCAR2LMNACYP11B2CYP11B1CYP1A2
SCHEMBL31032288 0.79 HCAR2 (0.49) HCAR2ALDH1A1KDM4EMEN1KMT2A
SCHEMBL30610133 0.79 HCAR2 (0.49) HCAR2ALDH1A1KDM4EMEN1KMT2A
SCHEMBL3942208 0.79 HCAR2 (0.49) HCAR2ALDH1A1KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116710430-A Methods and compounds for restoring mutant p53 function 皮姆维制药公司 2023-09-05 CN disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed