SCHEMBL10176215

SCHEMBL10176215

Cn1c(-c2ccncc2Cl)nc2cc(Cl)c(Cl)cc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KDM4E B2RXH2 3/20 0.42
LMNA P02545 1/20 0.42
ATM Q13315 1/20 0.42
PDE2A O00408 3/20 0.40
PDE10A Q9Y233 3/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
KCNH2 Q12809 1/20 0.40
AOC3 Q16853 1/20 0.40
PTPN1 P18031 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
HPGD P15428 1/20 0.39
CYP19A1 P11511 1/20 0.38
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
CASP1 P29466 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896741 0.89 CYP11B2 (0.47) POLBSMN1; SMN2KDM4EATMPDE2A
SCHEMBL17896660 0.87 CYP11B2 (0.43) POLBSMN1; SMN2KDM4ELMNAATM
SCHEMBL10248939 0.86 AGPAT2 (0.50) POLBSMN1; SMN2KDM4ELMNAATM
SCHEMBL10175361 0.86 PDE2A (0.52) POLBSMN1; SMN2KDM4EATMPDE2A
SCHEMBL10175127 0.83 CYP11B2 (0.40) POLBSMN1; SMN2KDM4EATMPDE2A
SCHEMBL17896744 0.81 CYP11B2 (0.47) POLBSMN1; SMN2KDM4EATMCYP11B1
SCHEMBL17897061 0.80 CYP11B2 (0.45) POLBSMN1; SMN2LMNAPDE2APDE10A
SCHEMBL169419 0.80 AGPAT2 (0.48) POLBSMN1; SMN2ATMPDE2APDE10A
SCHEMBL17896659 0.80 MEN1 (0.59) SMN1; SMN2KDM4ELMNAATMCYP11B1
SCHEMBL17896663 0.78 CYP11B2 (0.56) CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed