SCHEMBL10176534

SCHEMBL10176534

Cc1ccc(C(C(=O)OC(C)(C)C)C(C)C(F)(F)F)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.38
XBP1 P17861 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
ACHE P22303 1/20 0.34
ALOX5 P09917 1/20 0.34
KEAP1 Q14145 1/20 0.34
NFE2L2 Q16236 1/20 0.34
AAK1 Q2M2I8 1/20 0.34
LMNA P02545 1/20 0.33
KMT2A Q03164 1/20 0.33
CA2 P00918 1/20 0.33
CTSL P07711 1/20 0.32
CTSB P07858 1/20 0.32
CTSS P25774 1/20 0.32
CTSK P43235 1/20 0.32
GPR119 Q8TDV5 1/20 0.32
ADRB2 P07550 1/20 0.32
ADRB1 P08588 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1178706 0.84 ALOX5 (0.41) APPXBP1TDP1AKR1C3AKR1C2
SCHEMBL11932087 0.83 KMT2A (0.40) TDP1AKR1C3AKR1C2ACHELMNA
SCHEMBL517023 0.83 KMT2A (0.40) TDP1AKR1C3AKR1C2ACHELMNA
SCHEMBL3696396 0.81 AAK1 (0.37) APPXBP1TDP1AKR1C3AKR1C2
SCHEMBL13471793 0.79 AKR1C3 (0.46) AKR1C3AKR1C2ACHEALOX5KEAP1
SCHEMBL6901052 0.79 AKR1C3 (0.46) AKR1C3AKR1C2ACHEALOX5KEAP1
SCHEMBL14798411 0.79 AKR1C3 (0.46) AKR1C3AKR1C2ACHEALOX5KEAP1
SCHEMBL14797744 0.79 AKR1C3 (0.46) AKR1C3AKR1C2ACHEALOX5KEAP1
SCHEMBL517260 0.79 CHRM2 (0.43) APPXBP1TDP1ACHEALOX5
SCHEMBL5215244 0.77 APP (0.49) APPXBP1TDP1AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120028971-A1 OXO-HETEROCYCLICALLY SUBSTITUTED ALKYL CARBOXYLIC ACIDS AND USE THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-02-02 US disclosed
US-20120028971-A1 OXO-HETEROCYCLICALLY SUBSTITUTED ALKYL CARBOXYLIC ACIDS AND USE THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-02-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120028971-A1 OXO-HETEROCYCLICALLY SUBSTITUTED ALKYL CARBOXYLIC ACIDS AND USE THEREOF AADAC, OTC, HCAR2 APP 4095/4885XBP1 3221/4885TDP1 2877/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.