SCHEMBL10178211

SCHEMBL10178211

N=C/C(=C\NC(CN)C(F)(F)F)c1cnn2c(-c3cccc(NC(=O)NCC(F)(F)F)c3)cnc2c1

nearest known ligand 0.52

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
FGFR3 P22607 20/20 0.52
KDR P35968 11/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10178625 0.91 FGFR3 (0.52) FGFR3KDR
SCHEMBL10177312 0.91 FGFR3 (0.55) FGFR3KDR
SCHEMBL10179722 0.89 FGFR3 (0.51) FGFR3KDR
SCHEMBL10178936 0.89 FGFR3 (0.55) FGFR3KDR
SCHEMBL10177416 0.89 FGFR3 (0.51) FGFR3KDR
SCHEMBL15984935 0.88 FGFR3 (0.52) FGFR3KDR
SCHEMBL15984920 0.88 FGFR3 (0.52) FGFR3KDR
SCHEMBL10181280 0.88 FGFR3 (0.49) FGFR3KDR
SCHEMBL15984924 0.87 FGFR3 (0.62) FGFR3KDR
SCHEMBL10177433 0.86 FGFR3 (0.50) FGFR3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012088266-A2 SUBSTITUTED IMIDAZOPYRIDAZINES AND BENZIMIDAZOLES AS INHIBITORS OF FGFR3 INCYTE CORPORATION (US) 2012-06-28 WO disclosed