SCHEMBL10180395

SCHEMBL10180395

CCCCOc1ccc(Cl)cc1C(=O)NCCc1ccc(-c2ccc(OC(=O)O)cc2Cl)cc1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.50
DNMT3A Q9Y6K1 1/20 0.50
HDAC1 Q13547 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
NLRP3 Q96P20 3/20 0.46
CNR2 P34972 2/20 0.46
AKR1C3 P42330 1/20 0.45
MCHR1 Q99705 1/20 0.45
TP53 P04637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10180958 0.92 DNMT3A (0.49) CNR1DNMT3AHDAC1HDAC6NLRP3
SCHEMBL10181010 0.92 DNMT3A (0.54) DNMT3AHDAC1HDAC6NLRP3CNR2
SCHEMBL10181141 0.91 DNMT3A (0.48) CNR1DNMT3AHDAC1HDAC6NLRP3
SCHEMBL10181758 0.90 DNMT3A (0.53) CNR1DNMT3AHDAC1HDAC6NLRP3
SCHEMBL10181170 0.89 DNMT3A (0.52) DNMT3AHDAC1HDAC6NLRP3CNR2
SCHEMBL10180483 0.89 DNMT3A (0.46) CNR1DNMT3AHDAC1HDAC6NLRP3
SCHEMBL10180948 0.89 DNMT3A (0.64) DNMT3AHDAC1HDAC6NLRP3
SCHEMBL10180600 0.89 DNMT3A (0.49) DNMT3AHDAC1HDAC6NLRP3AKR1C3
SCHEMBL1154747 0.88 PPARD (0.54) CNR1DNMT3AHDAC1HDAC6NLRP3
SCHEMBL10182164 0.88 NPC1 (0.48) CNR1DNMT3AHDAC1HDAC6NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2215065-B1 CCR10 ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2012-07-11 EP claimed