SCHEMBL1018061

SCHEMBL1018061

CN(CC=O)c1ccc2c(n1)CCN(CC(=O)N1CCN(C3CCC3)CC1)C2

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.36
ALDH1A1 P00352 5/20 0.35
KDM4E B2RXH2 4/20 0.35
ALOX15 P16050 1/20 0.35
HRH3 Q9Y5N1 6/20 0.34
KCNH2 Q12809 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
F10 P00742 1/20 0.34
TSHR P16473 2/20 0.33
KMT2A Q03164 2/20 0.33
PKM P14618 2/20 0.33
GAA P10253 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MTNR1B P49286 1/20 0.32
ENPP2 Q13822 1/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1016464 0.91 PARP1 (0.37) PARP1ALDH1A1KDM4EALOX15HRH3
SCHEMBL1070174 0.90 PARP1 (0.39) PARP1ALDH1A1KDM4EALOX15HRH3
SCHEMBL1603356 0.88 PARP1 (0.35) PARP1ALDH1A1KDM4EALOX15HRH3
SCHEMBL1018243 0.87 ADRA1A (0.41) PARP1ALDH1A1KDM4EHRH3HTT
SCHEMBL1018889 0.86 PARP1 (0.41) PARP1ALDH1A1KDM4EALOX15HRH3
SCHEMBL14420825 0.82 PARP1 (0.34) PARP1ALDH1A1KDM4EALOX15HRH3
SCHEMBL1017297 0.81 HRH3 (0.42) PARP1ALDH1A1KDM4EHRH3KCNH2
SCHEMBL1016304 0.81 HRH3 (0.43) PARP1ALDH1A1KDM4EHRH3KCNH2
SCHEMBL1016478 0.79 PARP1 (0.40) PARP1ALDH1A1KDM4EHRH3KCNH2
SCHEMBL1014079 0.79 HRH3 (0.41) PARP1ALDH1A1KDM4EALOX15HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1998620-B1 PIPERAZINYL OXOALKYL TETRAHYDROISOQUINOLINES AND RELATED ANALOGUES NEUROGEN CORP (US) 2011-01-12 EP disclosed