SCHEMBL10180907

SCHEMBL10180907

CN1CCCN(c2cnc3ccc(-c4ccc(O)cc4)cc3n2)CC1.Oc1ccc(-c2ccc3ncc(N4CCCN(CCc5ccccc5)CC4)nc3c2)cc1.Oc1ccc(-c2ccc3ncc(N4CCCN(Cc5ccccc5)CC4)nc3c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
CHKA P35790 5/20 0.47
HRH4 Q9H3N8 3/20 0.43
HTR3A P46098 1/20 0.43
CASP1 P29466 2/20 0.43
CASP5 P51878 2/20 0.43
CASP4 P49662 1/20 0.43
PIM2 Q9P1W9 1/20 0.42
MELK Q14680 1/20 0.42
EHMT2 Q96KQ7 1/20 0.42
MET P08581 3/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
POLB P06746 1/20 0.41
HCAR2 Q8TDS4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12812470 0.92 CASP1 (0.50) NPC1RAB9AHRH4HTR3ACASP1
SCHEMBL12812477 0.90 NPC1 (0.63) NPC1RAB9ACASP1CASP5CASP4
SCHEMBL12812480 0.89 NPC1 (0.53) NPC1RAB9AHRH4HTR3ACASP1
SCHEMBL12812478 0.87 NPC1 (0.68) NPC1RAB9ACASP1CASP5KDM4E
SCHEMBL12812474 0.84 HRH4 (0.54) HRH4HTR3AMETKDM4EALDH1A1
SCHEMBL10179187 0.84 CASP1 (0.47) NPC1RAB9AHRH4HTR3ACASP1
SCHEMBL1442598 0.83 NPC1 (0.51) NPC1RAB9APOLBHCAR2
SCHEMBL1443431 0.82 NPC1 (0.58) NPC1RAB9AHRH4HTR3ACASP1
SCHEMBL10180445 0.80 NPC1 (0.56) NPC1RAB9AHRH4CASP1CASP5
SCHEMBL1442666 0.80 HRH4 (0.59) HRH4HTR3AMETALDH1A1HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2473498-A1 SUBSTITUTED AMINOQUINOXALINES AS TYROSINE THREONINE KINASE INHIBITORS Bayer Pharma Aktiengesellschaft (DE) 2012-07-11 EP claimed