SCHEMBL10183070

SCHEMBL10183070

N#Cc1ccc2c(c1)CC(NS(=O)(=O)Nc1ccccc1)CN2Cc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FNTA P49354 17/20 0.55
FNTB P49356 17/20 0.55
HRAS P01112 1/20 0.42
KRAS P01116 1/20 0.42
PGGT1B P53609 1/20 0.42
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
THRB P10828 1/20 0.41
CACNA1G O43497 1/20 0.40
CACNA1H O95180 1/20 0.40
CACNA1I Q9P0X4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10182259 0.87 FNTA (0.54) FNTAFNTBHRASKRASPGGT1B
SCHEMBL648852 0.86 FNTA (0.71) FNTAFNTBMTNR1AMTNR1BTHRB
SCHEMBL653554 0.86 FNTA (0.71) FNTAFNTBMTNR1AMTNR1BTHRB
SCHEMBL648851 0.86 FNTA (0.71) FNTAFNTBMTNR1AMTNR1BTHRB
SCHEMBL650724 0.84 FNTA (0.55) FNTAFNTBHRASKRASPGGT1B
SCHEMBL12920276 0.84 FNTA (0.55) FNTAFNTBHRASKRASPGGT1B
SCHEMBL12894285 0.82 MTNR1A (0.41) FNTAFNTBMTNR1AMTNR1BCACNA1G
SCHEMBL652407 0.82 FNTA (0.51) FNTAFNTBHRASKRASPGGT1B
SCHEMBL651451 0.81 FNTA (0.67) FNTAFNTBTHRB
SCHEMBL651452 0.81 FNTA (0.67) FNTAFNTBTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119808-B2 Tetrahydroquinoline derivatives as cannabinoid receptor modulators BRISTOL-MYERS SQUIBB COMPANY (US) 2012-02-21 US disclosed
US-20110104315-A1 TETRAHYDROQUINOLINE DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS BRISTOL-MYERS SQUIBB COMPANY 2011-05-05 US disclosed
US-7884113-B2 Tetrahydroquinoline derivatives as cannabinoid receptor modulators BRISTOL-MYERS SQUIBB COMPANY (US) 2011-02-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110104315-A1 TETRAHYDROQUINOLINE DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS CNR2, CNR1, OPRL1 FNTA 1368/4885FNTB 2071/4885HRAS 3120/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.