SCHEMBL10187265

SCHEMBL10187265

Nc1ccc(OC2CCC2)cc1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 1/20 0.60
FURIN P09958 2/20 0.52
ALDH1A1 P00352 3/20 0.46
TDP1 Q9NUW8 3/20 0.46
TSHR P16473 2/20 0.46
CYP3A4 P08684 2/20 0.46
NFE2L2 Q16236 1/20 0.44
MAPK1 P28482 1/20 0.42
HRH1 P35367 2/20 0.42
BTK Q06187 1/20 0.42
HPGD P15428 1/20 0.40
TNK2 Q07912 2/20 0.40
MAOA P21397 1/20 0.39
ACACB O00763 3/20 0.39
HRH3 Q9Y5N1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL747626 0.95 PARP10 (0.55) PARP10FURINALDH1A1TDP1TSHR
SCHEMBL623629 0.93 PARP10 (0.53) PARP10FURINALDH1A1TDP1TSHR
SCHEMBL26012610 0.93 PARP10 (0.53) PARP10FURINALDH1A1TDP1TSHR
SCHEMBL8316329 0.91 FURIN (0.62) PARP10FURINALDH1A1TDP1TSHR
SCHEMBL6903727 0.90 TDP1 (0.50) PARP10FURINALDH1A1TDP1TSHR
SCHEMBL8314928 0.90 TDP1 (0.50) PARP10FURINALDH1A1TDP1TSHR
SCHEMBL2242868 0.82 PARP10 (0.55) PARP10FURINALDH1A1TSHRHRH1
SCHEMBL737639 0.81 HRH3 (0.63) HRH3
SCHEMBL17533980 0.81 HRH3 (0.58) HRH3
SCHEMBL6121373 0.80 HRH1 (0.68) PARP10HRH1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111100596-B Fluorine-containing polyimide binder, flexible metal laminated plate and preparation method thereof 东莞东阳光科研发有限公司 2021-11-12 CN claimed
CN-111876085-A Composite bonding sheet, flexible metal laminated board and preparation method thereof 东莞东阳光科研发有限公司 2020-11-03 CN claimed
CN-111100596-A Fluorine-containing polyimide binder, flexible metal laminated plate and preparation method thereof 东莞东阳光科研发有限公司 2020-05-05 CN claimed
EP-4676926-A1 BICYCLIC HETEROARYL COMPOUNDS FOR USE AS GPR35 MODULATORS ThirtyFiveBio Limited (GB) 2026-01-14 EP disclosed
WO-2024184650-A1 BICYCLIC HETEROARYL COMPOUNDS FOR USE AS GPR35 MODULATORS. ThirtyFiveBio Limited (GB) 2024-09-12 WO disclosed
WO-2024132001-A1 MULTITARGET NUCLEAR RECEPTOR LIGANDS BASED ON 2-(4-(QUINOLIN-2-YLOXY)PHENOXY)PROPANOIC ACID AND 2-(4-(QUINOXALIN-2-YLOXY)PHENOXY)PROPANOIC ACID FOR THE TREATMENT OF METABOLIC AND LIVER DISEASES CHARLES UNIVERSITY, FACULTY OF PHARMACY IN HRADEC KRALOVE (CZ) 2024-06-27 WO disclosed
CN-111876085-B Composite bonding sheet, flexible metal laminated board and preparation method thereof 东莞东阳光科研发有限公司 2022-09-27 CN disclosed
CN-113105475-B Inhibitors of bruton's tyrosine kinase and methods of use thereof 詹森药业有限公司 2022-09-09 CN disclosed
CN-111100596-B Fluorine-containing polyimide binder, flexible metal laminated plate and preparation method thereof 东莞东阳光科研发有限公司 2021-11-12 CN disclosed
CN-113105475-A Inhibitors of bruton's tyrosine kinase and methods of use thereof 詹森药业有限公司 2021-07-13 CN disclosed
US-10822348-B2 Inhibitors of Bruton's tyrosine kinase and methods of their use JANSSEN PHARMACEUTICA NV (BE) 2020-11-03 US disclosed
EP-3239150-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2020-02-05 EP disclosed
US-20190284203-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE AND METHOD OF THEIR USE JANSSEN PHARMACEUTICA NV (BE) 2019-09-19 US disclosed
US-20190284204-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE AND METHOD OF THEIR USE JANSSEN PHARMACEUTICA NV (BE) 2019-09-19 US disclosed
EP-2997024-B1 PYRROLIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF BOEHRINGER INGELHEIM INT (DE) 2018-03-28 EP disclosed
EP-3239150-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2017-11-01 EP disclosed
US-20170283431-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE AND METHOD OF THEIR USE JANSSEN PHARMACEUTICA NV (BE) 2017-10-05 US disclosed
EP-2797885-B1 NEW AZETIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF BOEHRINGER INGELHEIM INT (DE) 2016-08-10 EP disclosed
WO-2013079668-A1 PIPERIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-06-06 WO disclosed
WO-2012001107-A1 PIPERIDINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF METABOLIC DISORDERS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190284204-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE AND METHOD OF THEIR USE ABL1, BTK, MYLK2 PARP10 1392/4885FURIN 4155/4885ALDH1A1 4003/4885
US-10822348-B2 Inhibitors of Bruton's tyrosine kinase and methods of their use ABL1, BTK, MYLK2 PARP10 1231/4885FURIN 4127/4885ALDH1A1 3899/4885
US-20170283431-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE AND METHOD OF THEIR USE ABL1, BTK, MYLK2 PARP10 1392/4885FURIN 4155/4885ALDH1A1 4003/4885
US-20190284203-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE AND METHOD OF THEIR USE ABL1, BTK, MYLK2 PARP10 1392/4885FURIN 4155/4885ALDH1A1 4003/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.