SCHEMBL10187278

SCHEMBL10187278

CC(C)[C@@H](C)Nc1cc(N)ncn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.39
CCNB1 P14635 1/20 0.39
CCNA2 P20248 1/20 0.39
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39
CDK5 Q00535 1/20 0.39
CDK5R1 Q15078 1/20 0.39
PIK3CD O00329 2/20 0.38
PIK3R1 P27986 2/20 0.38
SCN9A Q15858 1/20 0.37
KDR P35968 1/20 0.37
HCAR3 P49019 1/20 0.37
MKNK2 Q9HBH9 1/20 0.35
IDH1 O75874 1/20 0.35
MAPK14 Q16539 6/20 0.35
CA2 P00918 1/20 0.34
CHKA P35790 1/20 0.34
HRH4 Q9H3N8 1/20 0.34
JAK2 O60674 1/20 0.33
JAK3 P52333 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17591565 0.84 JAK2 (0.43) CDK1CCNB1CCNA2CCNE1CDK2
SCHEMBL30579411 0.84 JAK2 (0.43) CDK1CCNB1CCNA2CCNE1CDK2
SCHEMBL18815015 0.77 NPC1 (0.42) HCAR3MAPK14MEN1KMT2A
SCHEMBL23024945 0.77 LRRK2 (0.39) CDK1CCNB1CCNA2CCNE1CDK2
SCHEMBL23024921 0.77 LRRK2 (0.39) CDK1CCNB1CCNA2CCNE1CDK2
SCHEMBL30047569 0.74 HTR7 (0.58) PIK3CDPIK3R1MAPK14JAK2JAK3
SCHEMBL23059301 0.73 MEN1 (0.42) PIK3CDPIK3R1HCAR3IDH1CA2
SCHEMBL23059377 0.73 MEN1 (0.42) PIK3CDPIK3R1HCAR3IDH1CA2
SCHEMBL1911881 0.73
SCHEMBL29741837 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012001107-A1 PIPERIDINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF METABOLIC DISORDERS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-05 WO disclosed